SCHEMBL7863294

SCHEMBL7863294

NC(=S)Nc1cccc(S(=O)(=O)Nc2cccc(CC(C(=O)O)c3ccccc3)c2)c1

nearest known ligand 0.48

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HTR6 P50406 6/20 0.48
PTGES O14684 1/20 0.43
ALDH1A1 P00352 2/20 0.43
PKM P14618 2/20 0.43
CA1 P00915 5/20 0.42
CA2 P00918 5/20 0.42
CA9 Q16790 4/20 0.42
CA12 O43570 3/20 0.42
L3MBTL1 Q9Y468 1/20 0.42
MAPT P10636 2/20 0.41
NAMPT P43490 1/20 0.41
ITGB3 P05106 1/20 0.41
ITGAV P06756 1/20 0.41
MEN1 O00255 1/20 0.41
LMNA P02545 1/20 0.41
MAPK1 P28482 1/20 0.41
KMT2A Q03164 1/20 0.41
NOS3 P29474 1/20 0.40
NOS1 P29475 1/20 0.40
NOS2 P35228 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7856532 0.92 CA1 (0.51) HTR6PTGESALDH1A1PKMCA1
SCHEMBL7861976 0.87 CA12 (0.43) HTR6PTGESALDH1A1PKMCA1
SCHEMBL7864272 0.86 NAMPT (0.58) HTR6CA1CA2CA9CA12
SCHEMBL7863291 0.80 ITGB3 (0.45) HTR6PKMCA1CA2CA9
SCHEMBL7861846 0.79 CA1 (0.44) HTR6PTGESALDH1A1PKMCA1
SCHEMBL7856518 0.79 PTGES (0.40) HTR6PTGESALDH1A1PKMCA1
SCHEMBL6366661 0.77 GBA1 (0.46) HTR6ALDH1A1PKMCA1CA2
SCHEMBL31689529 0.74 HTR6 (0.64) HTR6PTGESPKMMEN1KMT2A
SCHEMBL7861972 0.74 TGFBR1 (0.43) ALDH1A1PKMCA1CA2MAPT
SCHEMBL7864224 0.74 NAMPT (0.51) ALDH1A1CA1CA2CA9CA12

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0889877-B1 META-SUBSTITUTED PHENYLENE DERIVATIVES AND THEIR USE AS ALPHAvBETA3 INTEGRIN ANTAGONISTS OR INHIBITORS SEARLE & CO (US) 2001-08-29 EP claimed