SCHEMBL78635

SCHEMBL78635

CCC1=C(c2cccc(-c3ccccc3)c2)CC(CO[Si](C)(C)C(C)(C)C)N(C(=O)OCc2ccccc2)C1

nearest known ligand 0.37

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PDK1 Q15118 1/20 0.35
PDK2 Q15119 1/20 0.35
PDK3 Q15120 1/20 0.35
PDK4 Q16654 1/20 0.35
TMEM97 Q5BJF2 2/20 0.34
SIGMAR1 Q99720 2/20 0.34
NPSR1 Q6W5P4 1/20 0.34
MGLL Q99685 1/20 0.34
CHRM2 P08172 1/20 0.33
CHRM4 P08173 1/20 0.33
CHRM5 P08912 1/20 0.33
CHRM1 P11229 1/20 0.33
CHRM3 P20309 1/20 0.33
HDAC1 Q13547 1/20 0.33
HDAC2 Q92769 1/20 0.33
HTR2C P28335 1/20 0.33
KDM4E B2RXH2 1/20 0.33
NPC1 O15118 1/20 0.33
ALDH1A1 P00352 1/20 0.33
RAB9A P51151 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL65202 0.90 MGLL (0.36) PDK1PDK2PDK3PDK4TMEM97
SCHEMBL78404 0.90 PDK1 (0.35) PDK1PDK2PDK3PDK4TMEM97
SCHEMBL65231 0.88 CHRM5 (0.39) PDK1PDK2PDK3PDK4TMEM97
SCHEMBL78366 0.87 PDK1 (0.33) PDK1PDK2PDK3PDK4NPSR1
SCHEMBL78724 0.82 KDM4E (0.34) CHRM5CHRM1KDM4E
SCHEMBL78854 0.81 PPARG (0.40) KDM4EALDH1A1SMN1; SMN2
SCHEMBL8701755 0.80 PSEN1 (0.41) PDK1PDK2PDK3PDK4NPSR1
SCHEMBL8701756 0.80 PSEN1 (0.41) PDK1PDK2PDK3PDK4NPSR1
SCHEMBL64061 0.80 CHRM2 (0.38) PDK1PDK2PDK3PDK4TMEM97
SCHEMBL78407 0.80 PDK1 (0.37) PDK1PDK2PDK3PDK4HTR2C

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-8129538-B1 Renin inhibitors TAKEDA PHARMACEUTICAL COMPANY LIMITED (JP) 2012-03-06 US disclosed