SCHEMBL7863517

SCHEMBL7863517

CC(C)(C)OC(=O)N1CCC(CCCn2c(=O)c3cnc4cccc2n43)CC1

nearest known ligand 0.46

Predicted protein targets (top 8)

geneUniProtsupporting neighboursconfidence
GPR119 Q8TDV5 11/20 0.46
FAAH O00519 1/20 0.45
SGMS2 Q8NHU3 5/20 0.44
SGMS1 Q86VZ5 4/20 0.44
KDM4E B2RXH2 1/20 0.42
PKM P14618 1/20 0.42
PIK3CA P42336 1/20 0.41
PRKDC P78527 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7871693 0.95 GPR119 (0.43) GPR119FAAHSGMS2SGMS1KDM4E
SCHEMBL7863410 0.91 PIK3CA (0.46) GPR119FAAHKDM4EPKMPIK3CA
SCHEMBL7868718 0.84 PIK3CA (0.46) GPR119FAAHSGMS2SGMS1KDM4E
SCHEMBL8712463 0.83 GPR119 (0.43) GPR119FAAHKDM4EPKM
SCHEMBL7871606 0.79 GPR119 (0.45) GPR119FAAHKDM4EPKM
SCHEMBL7863491 0.77 GPR119 (0.45) GPR119FAAHKDM4EPKM
SCHEMBL8713112 0.74 GPR119 (0.45) GPR119FAAHKDM4EPKM
SCHEMBL7863430 0.74 GPR119 (0.46) GPR119FAAHKDM4EPKM
SCHEMBL7868708 0.74 GPR119 (0.43) GPR119KDM4EPKMPIK3CAPRKDC
SCHEMBL948301 0.73 GPR119 (0.48) GPR119KDM4E

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20010051631-A1 Tricyclic compounds, their production and use TAKATANI MUNEO (JP) 2001-12-13 US disclosed
US-6251905-B1 Tricyclic compounds, their production and use TAKEDA CHEMICAL INDUSTRIES, LTD. (JP) 2001-06-26 US disclosed
EP-0826686-A2 Tricyclic compounds, their production and use TAKEDA CHEMICAL INDUSTRIES, LTD. (JP) 1998-03-04 EP disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20010051631-A1 Tricyclic compounds, their production and use PDGFA, HGF, REN GPR119 605/4885FAAH 1223/4885SGMS2 647/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.