SCHEMBL7866630

SCHEMBL7866630

CNCCc1c[nH]c2ccc(NC(=O)c3ccc(F)cc3)cc12

nearest known ligand 0.64

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MPO P05164 2/20 0.64
SNCA P37840 3/20 0.58
SIRT1 Q96EB6 1/20 0.56
MAPT P10636 1/20 0.55
HTR1D P28221 5/20 0.55
HTR1B P28222 3/20 0.55
HTR1A P08908 2/20 0.55
KDM4E B2RXH2 2/20 0.55
MTNR1A P48039 2/20 0.55
MTNR1B P49286 2/20 0.55
NOTUM Q6P988 2/20 0.55
ALDH1A1 P00352 1/20 0.55
LMNA P02545 1/20 0.55
NPSR1 Q6W5P4 1/20 0.55
TDP1 Q9NUW8 1/20 0.55
HTR1F P30939 1/20 0.54
MEN1 O00255 1/20 0.54
CYP2D6 P10635 1/20 0.54
HTR2C P28335 1/20 0.54
KMT2A Q03164 1/20 0.54

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Water SCHEMBL10579379 0.80 KDM4E (0.60) MPOMAPTHTR1DHTR1BHTR1A
SCHEMBL7141265 0.79 HTR1F (0.76) SNCAMAPTHTR1DHTR1BHTR1A
SCHEMBL2404396 0.79 MPO (1.00) MPOHTR1DHTR1BHTR1AKDM4E
SCHEMBL7860320 0.78 HTR1F (0.50) MPOMAPTHTR1DHTR1BHTR1A
SCHEMBL9256341 0.78 MPO (0.53) MPOSNCASIRT1MAPTHTR1D
SCHEMBL12352653 0.77 KDM4E (0.70) MPOMAPTHTR1DHTR1BHTR1A
SCHEMBL7860323 0.76 MMP2 (0.49) HTR1DHTR1BHTR1AHTR1FMEN1
SCHEMBL11359819 0.76 HTR1A (0.71) MPOMAPTHTR1DHTR1BHTR1A
SCHEMBL20182262 0.76 TRPV1 (0.73) SNCASIRT1MAPTKDM4EMTNR1A
Hydrochloric Acid SCHEMBL8194413 0.76 HTR1F (0.47) MPOSNCAMAPTHTR1DHTR1B

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1083918-A1 NOVEL THERAPEUTIC AGENTS THAT MODULATE 5-HT RECEPTORS Advanced Medicine, Inc. (US) 2001-03-21 EP disclosed
WO-1999064044-A1 NOVEL THERAPEUTIC AGENTS THAT MODULATE 5-HT RECEPTORS ADVANCED MEDICINE, INC. (US) 1999-12-16 WO disclosed