SCHEMBL7869467

SCHEMBL7869467

COCCNC(=O)Oc1ccc(C(=O)NS(=O)(=O)c2ccc(NC(=O)Cc3ccccc3)cc2)cn1

nearest known ligand 0.48

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MEN1 O00255 2/20 0.48
KMT2A Q03164 2/20 0.48
SCN3A Q9NY46 1/20 0.45
LMNA P02545 3/20 0.45
BCL2 P10415 1/20 0.45
BCL2L1 Q07817 1/20 0.45
MCL1 Q07820 1/20 0.45
NPC1 O15118 2/20 0.44
RAB9A P51151 1/20 0.44
PKM P14618 2/20 0.44
PRMT1 Q99873 1/20 0.43
NAMPT P43490 1/20 0.43
PPARA Q07869 1/20 0.43
KDM4E B2RXH2 1/20 0.43
BDKRB1 P46663 1/20 0.43
L3MBTL1 Q9Y468 1/20 0.43
RORC P51449 1/20 0.42
CA12 O43570 1/20 0.42
CA1 P00915 1/20 0.42
CA2 P00918 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9574752 0.92 L3MBTL1 (0.53) MEN1KMT2ALMNABCL2BCL2L1
SCHEMBL7870480 0.91 SCN3A (0.46) MEN1KMT2ASCN3ALMNABCL2
SCHEMBL7862672 0.91 L3MBTL1 (0.47) MEN1KMT2ALMNABCL2BCL2L1
SCHEMBL9574869 0.90 CA1 (0.47) MEN1KMT2ABCL2L1MCL1NPC1
SCHEMBL7862839 0.90 SMN1; SMN2 (0.48) LMNAPKMNAMPTPPARAKDM4E
SCHEMBL9574735 0.89 ALDH1A1 (0.52) MEN1KMT2ALMNAPKM
SCHEMBL7869445 0.89 PKM (0.43) MEN1KMT2APKMNAMPTKDM4E
SCHEMBL9018559 0.88 MEN1 (0.53) MEN1KMT2ASCN3ALMNANPC1
SCHEMBL7871609 0.87 P4HTM (0.55) BCL2L1MCL1NAMPTP4HTM
SCHEMBL8868481 0.87 HDAC3 (0.51) MEN1KMT2ASCN3ALMNABCL2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0562512-B1 Sulfonamidocarbonylpyridine-2-carboxamides and their use as medicines HOECHST AG (DE) 2001-02-21 EP disclosed
EP-0562512-A1 Sulfonamido- and sulfonamidocarbonyl-pyridine-2-carboxamides and their pyridine-N-oxides, process for their preparation and their use as medicines HOECHST AKTIENGESELLSCHAFT (DE) 1993-09-29 EP disclosed