SCHEMBL7874401

SCHEMBL7874401

COc1c[c]c(-c2ccc(C(F)(F)F)cc2)c(OC)c1OC

nearest known ligand 0.42

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
SMN1; SMN2 Q16637 2/20 0.42
RAB9A P51151 2/20 0.42
NPSR1 Q6W5P4 1/20 0.42
NFE2L2 Q16236 1/20 0.40
ALDH1A1 P00352 1/20 0.39
HPGD P15428 1/20 0.39
KIF11 P52732 6/20 0.38
AKR1C3 P42330 1/20 0.36
AKR1C2 P52895 1/20 0.36
BCL9 O00512 1/20 0.36
CTNNB1 P35222 1/20 0.36
ALOX5AP P20292 1/20 0.36
FEN1 P39748 1/20 0.36
IDO1 P14902 1/20 0.36
TDO2 P48775 1/20 0.36
TSHR P16473 1/20 0.35
CASR P41180 2/20 0.35
TNKS O95271 1/20 0.35
TNKS2 Q9H2K2 1/20 0.35
PARP2 Q9UGN5 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL28334181 0.80 CA12 (0.39) ALDH1A1IDO1TDO2
SCHEMBL14775511 0.79 LMNA (0.36) NPSR1TSHRMAPT
SCHEMBL7699767 0.78 KDM4E (0.39) SMN1; SMN2NFE2L2ALDH1A1HPGDIDO1
SCHEMBL9509766 0.76 TUBB4A (0.43) SMN1; SMN2RAB9AALDH1A1HPGDTSHR
SCHEMBL9738424 0.73 ACHE (0.43) SMN1; SMN2ALDH1A1HPGDTSHRKDM4E
SCHEMBL9538022 0.72 MAOB (0.44) ALDH1A1KDM4EMAPT
SCHEMBL14450971 0.71 KIF11 (0.52) SMN1; SMN2RAB9ANPSR1NFE2L2ALDH1A1
SCHEMBL6575991 0.68 MAPK1 (0.48) SMN1; SMN2RAB9AALDH1A1KDM4ECYP1A2
SCHEMBL3294513 0.67 AKR1C3 (0.56) SMN1; SMN2RAB9ANPSR1KIF11AKR1C3
SCHEMBL1133231 0.66 AR (0.53) SMN1; SMN2RAB9ANPSR1NFE2L2HPGD

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0754176-B1 NOVEL CARBAMATES AND UREAS AS MODIFIERS OF MULTI-DRUG RESISTANCE VERTEX PHARMA (US) 2001-12-05 EP claimed