SCHEMBL7876520

SCHEMBL7876520

C[C@@H]([C@@H](CC1CCCc2ccccc21)C(=O)O)N(O)C=O

nearest known ligand 0.42

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 3/20 0.42
HTT P42858 4/20 0.40
XBP1 P17861 1/20 0.40
KDM4C Q9H3R0 4/20 0.39
KDM5A P29375 2/20 0.39
KDM5B Q9UGL1 2/20 0.39
RAB9A P51151 1/20 0.39
BLM P54132 1/20 0.39
TSHR P16473 1/20 0.39
MEN1 O00255 1/20 0.38
KMT2A Q03164 1/20 0.38
FFAR1 O14842 1/20 0.37
HTR6 P50406 1/20 0.37
PDPK1 O15530 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7873347 0.76 CA2 (0.40)
SCHEMBL5951346 0.75 TSHR (0.47) ALDH1A1HTTXBP1KDM4CKDM5A
SCHEMBL7876518 0.73 MAPK1 (0.42) ALDH1A1HTTXBP1RAB9ABLM
SCHEMBL14632819 0.72 CYP19A1 (0.45) ALDH1A1HTTXBP1PDPK1
SCHEMBL3590904 0.72 FFAR1 (0.52) ALDH1A1HTTXBP1KDM4CKDM5A
SCHEMBL30301824 0.72 FFAR1 (0.52) ALDH1A1HTTXBP1KDM4CKDM5A
SCHEMBL6541484 0.71 PRCP (0.53) ALDH1A1
SCHEMBL9683763 0.70 BLM (0.50) ALDH1A1HTTXBP1KDM4CKDM5A
SCHEMBL2995330 0.69 CHRM1 (0.43) PDPK1
SCHEMBL7038866 0.69 HAO1 (0.53) ALDH1A1HTTXBP1KDM4CKDM5A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6329400-B1 INHIBITION OR ANTAGONISM OF MATRIX METALLOPROTEASES, AND/OR TUMOR NECROSIS FACTOR-ALPHA; EXTRACELLULAR MATRIX DEGRADATION, INHIBITION OF SHEDDING OF CELL SURFACE PROTEIN ECTODOMAINS AND CD23 PROTEOLYSIS GLAXO WELLCOME INC. 2001-12-11 US disclosed