SCHEMBL78858

SCHEMBL78858

CCC1CN(C(=O)OCc2ccccc2)C(CO[Si](C)(C)C(C)(C)C)C=C1c1ccc(OCCOc2ccccc2Cl)cc1

nearest known ligand 0.40

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PPARA Q07869 6/20 0.40
PPARD Q03181 4/20 0.40
PPARG P37231 3/20 0.40
KDM4E B2RXH2 2/20 0.34
LMNA P02545 1/20 0.34
L3MBTL1 Q9Y468 3/20 0.33
S1PR5 Q9H228 2/20 0.33
S1PR1 P21453 1/20 0.33
PRKX P51817 1/20 0.33
ACVR1 Q04771 1/20 0.33
TSHR P16473 1/20 0.32
SMN1; SMN2 Q16637 2/20 0.32
PDK1 Q15118 1/20 0.32
PDK2 Q15119 1/20 0.32
PDK3 Q15120 1/20 0.32
PDK4 Q16654 1/20 0.32
NPC1 O15118 1/20 0.32
RAB9A P51151 1/20 0.32
MEN1 O00255 1/20 0.32
ALDH1A1 P00352 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL78725 0.93 KDM4E (0.34) PPARAPPARDPPARGKDM4ELMNA
SCHEMBL78706 0.88 PPARA (0.37) PPARAPPARDPPARGKDM4ELMNA
SCHEMBL78419 0.81 PDK1 (0.32) PPARGKDM4ELMNAS1PR5S1PR1
SCHEMBL78854 0.80 PPARG (0.40) PPARAPPARDPPARGKDM4ELMNA
SCHEMBL91347 0.80 PPARG (0.38) PPARAPPARDPPARGKDM4ELMNA
SCHEMBL65792 0.79 PPARA (0.39) PPARAPPARDPPARGKDM4ELMNA
SCHEMBL64456 0.79 PPARG (0.39) PPARAPPARDPPARGKDM4ELMNA
SCHEMBL78412 0.78 PPARG (0.39) PPARAPPARDPPARGKDM4ELMNA
SCHEMBL64056 0.78 PPARG (0.38) PPARAPPARDPPARGKDM4ELMNA
SCHEMBL64057 0.77 PPARG (0.39) PPARAPPARDPPARGKDM4ELMNA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-8129538-B1 Renin inhibitors TAKEDA PHARMACEUTICAL COMPANY LIMITED (JP) 2012-03-06 US disclosed