SCHEMBL78419

SCHEMBL78419

CC(C)(C)[Si](C)(C)OCC1C=C(c2ccc(OCCOc3c(Cl)cccc3Cl)cc2)C(OC=O)CN1C(=O)OCc1ccccc1

nearest known ligand 0.34

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
PDK1 Q15118 1/20 0.32
PDK2 Q15119 1/20 0.32
PDK3 Q15120 1/20 0.32
PDK4 Q16654 1/20 0.32
KDM4E B2RXH2 1/20 0.31
LMNA P02545 1/20 0.31
FFAR2 O15552 1/20 0.31
PPARG P37231 1/20 0.31
S1PR5 Q9H228 2/20 0.31
S1PR1 P21453 1/20 0.31
PRKX P51817 1/20 0.31
ACVR1 Q04771 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL78706 0.93 PPARA (0.37) PDK1PDK2PDK3PDK4KDM4E
SCHEMBL78725 0.88 KDM4E (0.34) PDK1PDK2PDK3PDK4KDM4E
SCHEMBL78858 0.81 PPARA (0.40) PDK1PDK2PDK3PDK4KDM4E
SCHEMBL80037 0.79 ITGB3 (0.32) KDM4ELMNAFFAR2
SCHEMBL64503 0.78 PPARA (0.33) KDM4ELMNAPPARG
SCHEMBL10289281 0.78 FABP4 (0.34) PDK1PDK2PDK3PDK4KDM4E
SCHEMBL64196 0.77 GHSR (0.36) KDM4ELMNA
SCHEMBL78724 0.77 KDM4E (0.34) KDM4ELMNAPPARG
SCHEMBL64233 0.76 CHRM5 (0.35) KDM4ELMNA
SCHEMBL10289283 0.76 KDM4E (0.33) KDM4ELMNA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-8129538-B1 Renin inhibitors TAKEDA PHARMACEUTICAL COMPANY LIMITED (JP) 2012-03-06 US disclosed