SCHEMBL7898720

SCHEMBL7898720

N=C(N)Nc1cccc(CBr)c1

nearest known ligand 0.43

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
ITGB3 P05106 1/20 0.43
ITGA2B P08514 1/20 0.43
SIGMAR1 Q99720 11/20 0.42
GRIN2D O15399 3/20 0.42
GRIN3B O60391 3/20 0.42
GRIN1 Q05586 3/20 0.42
GRIN2A Q12879 3/20 0.42
GRIN2B Q13224 3/20 0.42
GRIN2C Q14957 3/20 0.42
GRIN3A Q8TCU5 3/20 0.42
SLC11A2 P49281 1/20 0.38
NOS3 P29474 1/20 0.38
NOS1 P29475 1/20 0.38
NOS2 P35228 1/20 0.38
PARP1 P09874 1/20 0.37
PLAU P00749 1/20 0.37
NPSR1 Q6W5P4 1/20 0.37
KMT2A Q03164 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6678310 0.84 LOXL2 (0.55) ITGB3ITGA2BSIGMAR1GRIN2DGRIN3B
SCHEMBL28347492 0.84 ITGB3 (0.43) ITGB3ITGA2BSIGMAR1GRIN2DGRIN3B
[3-(Hydroxymethyl)Phenyl]Guanidine SCHEMBL1186272 0.84 PRSS1 (0.55) ITGB3ITGA2BSIGMAR1GRIN2DGRIN3B
SCHEMBL5212905 0.82 MAPT (0.46) ITGB3ITGA2BSIGMAR1GRIN2DGRIN3B
SCHEMBL8432263 0.82 ITGB3 (0.46) ITGB3ITGA2BSIGMAR1GRIN2DGRIN3B
Hydrochloric Acid SCHEMBL6680642 0.82 LOXL2 (0.53) ITGB3ITGA2BSIGMAR1GRIN2DGRIN3B
SCHEMBL8269124 0.82 SIGMAR1 (0.60) SIGMAR1GRIN2DGRIN3BGRIN1GRIN2A
SCHEMBL3728364 0.81 NOS1 (0.50) ITGB3ITGA2BSIGMAR1GRIN2DGRIN3B
SCHEMBL14470096 0.81 ITGB3 (0.42) ITGB3ITGA2BSIGMAR1GRIN2DGRIN3B
SCHEMBL1184796 0.81 SIRT1 (0.51) ITGB3ITGA2BSIGMAR1GRIN2DGRIN3B

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6191273-B1 3,6,10,14-SUBSTITUTED-3,6,10,16-TETRAAZABICYCLO(10.3.1)-HEXADE CA-1(16),12,14-TRIENE COMPOUNDS OF GIVEN FORMULA; ANTIBACTERIAL AND OTHER UTILITIES, SUCH AS TO SCREEN FOR PESTICIDES OR DRUGS ISIS PHARMACEUTICALS, INC. 2001-02-20 US disclosed
WO-1999011612-A2 SUBSTITUTED CYCLIC COMPOUNDS AND MIXTURES COMPRISING SAME ISIS PHARMACEUTICALS, INC. (US) 1999-03-11 WO disclosed