SCHEMBL7900907

SCHEMBL7900907

COC(=O)c1ccc(OCCc2c[nH]c3ccccc23)cc1O

nearest known ligand 0.55

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PTGS1 P23219 3/20 0.54
NR4A2 P43354 1/20 0.52
CREBBP Q92793 1/20 0.52
PTGS2 P35354 2/20 0.52
GPR84 Q9NQS5 1/20 0.51
SIRT1 Q96EB6 1/20 0.51
CDK2 P24941 2/20 0.51
MTNR1A P48039 2/20 0.51
MTNR1B P49286 2/20 0.51
MAPT P10636 4/20 0.50
MEN1 O00255 3/20 0.50
KMT2A Q03164 3/20 0.50
NPC1 O15118 1/20 0.50
POLB P06746 1/20 0.50
RAB9A P51151 1/20 0.50
LTA4H P09960 1/20 0.49
PLA2G2A P14555 1/20 0.49
ALDH1A1 P00352 1/20 0.49
LMNA P02545 1/20 0.49
SMN1; SMN2 Q16637 1/20 0.49

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7911142 0.88 MTNR1A (0.53) CDK2MTNR1AMTNR1BMAPTMEN1
SCHEMBL6516526 0.84 GPR84 (0.61) GPR84CDK2MAPTMEN1KMT2A
SCHEMBL5116952 0.81 MAOA (0.60) MAPTMEN1KMT2ANPC1POLB
SCHEMBL7901014 0.78 MAOB (0.57) MAPTMEN1KMT2APOLBLMNA
SCHEMBL7911137 0.78 ALDH1A1 (0.53) CDK2MTNR1AMTNR1BMAPTMEN1
SCHEMBL8998953 0.78 EGFR (0.67) PTGS1PTGS2MAPTMEN1KMT2A
SCHEMBL6516758 0.77 MAPT (0.57) MTNR1AMTNR1BMAPTMEN1KMT2A
SCHEMBL6516295 0.76 MAPT (0.60) MTNR1AMTNR1BMAPTMEN1KMT2A
SCHEMBL4800518 0.76 NR4A2 (0.46) NR4A2CREBBPMTNR1AMTNR1BMAPT
SCHEMBL11461356 0.76 PPARD (0.59) MAPTNPC1POLBRAB9APLA2G2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6211234-B1 BENZONITRILE COMPOUNDS WITH ETHER AND SULFIDE GROUPS WITH CARBOXY ACID RHONE-POULENC RORER LIMITED (GB) 2001-04-03 US disclosed
EP-0728128-B1 SUBSTITUTED PHENYL COMPOUNDS RHONE POULENC RORER LTD (GB) 1998-09-16 EP disclosed
EP-0728128-A1 SUBSTITUTED PHENYL COMPOUNDS RHONE-POULENC RORER LIMITED (GB) 1996-08-28 EP disclosed
WO-1995013262-A1 SUBSTITUTED PHENYL COMPOUNDS RHONE-POULENC RORER LIMITED (GB) 1995-05-18 WO disclosed