SCHEMBL7902606

SCHEMBL7902606

CSc1nc(N)n(-c2nnc(-c3ccccc3OCCBr)s2)n1

nearest known ligand 0.36

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KDM4E B2RXH2 4/20 0.36
ALDH1A1 P00352 3/20 0.36
HRH3 Q9Y5N1 1/20 0.32
HSD17B10 Q99714 3/20 0.32
HPGD P15428 2/20 0.32
NPC1 O15118 1/20 0.31
LMNA P02545 1/20 0.31
RAB9A P51151 1/20 0.31
MEN1 O00255 1/20 0.31
POLB P06746 1/20 0.31
MAPT P10636 1/20 0.31
TSHR P16473 1/20 0.31
KMT2A Q03164 1/20 0.31
NPSR1 Q6W5P4 1/20 0.31
CA12 O43570 1/20 0.31
CA1 P00915 1/20 0.31
CA2 P00918 1/20 0.31
CA9 Q16790 1/20 0.31
MGAM O43451 1/20 0.30
GAA P10253 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7902622 0.95 KDM4E (0.36) KDM4EALDH1A1HRH3HSD17B10HPGD
SCHEMBL7904668 0.88 ALDH1A1 (0.37) KDM4EALDH1A1
SCHEMBL7896441 0.87 HTR1B (0.37) KDM4EALDH1A1HRH3
SCHEMBL7903994 0.87 ATP4A (0.40) HRH3
SCHEMBL7896514 0.85 HRH3 (0.42) KDM4EALDH1A1HRH3LMNAMEN1
SCHEMBL7903985 0.84 KDM4E (0.34) KDM4EALDH1A1HRH3HSD17B10HPGD
SCHEMBL7904663 0.84 MEN1 (0.35) KDM4EALDH1A1HRH3LMNAMEN1
SCHEMBL7896411 0.83 USP2 (0.43) KDM4EALDH1A1HRH3LMNAPOLB
SCHEMBL7904676 0.82 RAB9A (0.33) KDM4EALDH1A1HSD17B10HPGDNPC1
SCHEMBL7904717 0.81 MAOB (0.33) KDM4EALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6191152-B1 CARDIOVASCULAR DISORDERS, NERVOUS SYSTEM DISORDERS EGIS GYÓGYSZERGYAR RT. (HU) 2001-02-20 US disclosed
EP-0958294-A1 2-(1,2,4-TRIAZOLE-1-YL)-1,3,4-THIADIAZOLE DERIVATIVES HAVING AN EFFECT ON THE C.N.S. AND THE HEART EGIS GYOGYSZERGYAR (HU) 1999-11-24 EP disclosed
WO-1998030561-A1 2-(1,2,4-TRIAZOLE-1-YL)-1,3,4-THIADIAZOLE DERIVATIVES HAVING AN EFFECT ON THE C.N.S. AND THE HEART EGIS Gyógyszergyár Rt. (HU) 1998-07-16 WO disclosed