SCHEMBL790553

SCHEMBL790553

Nc1nc2ccc(-c3cncc(NC(=O)c4ccccc4)c3)cc2cc1-c1ccc(N2CCOCC2)cc1

nearest known ligand 0.49

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ATR Q13535 2/20 0.49
TP53 P04637 1/20 0.46
SMN1; SMN2 Q16637 1/20 0.46
MAPK1 P28482 1/20 0.46
PI4KA P42356 1/20 0.46
PIK3CG P48736 1/20 0.46
MAPT P10636 2/20 0.45
ROCK1 Q13464 1/20 0.45
DGAT1 O75907 2/20 0.44
JAK2 O60674 1/20 0.44
JAK1 P23458 1/20 0.44
TYK2 P29597 1/20 0.44
JAK3 P52333 1/20 0.44
MAPK14 Q16539 1/20 0.44
RPS6KA2 Q15349 1/20 0.43
HDAC3 O15379 1/20 0.43
HDAC4 P56524 1/20 0.43
HDAC1 Q13547 1/20 0.43
HDAC7 Q8WUI4 1/20 0.43
HDAC2 Q92769 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL790788 0.91 NPC1 (0.54) ATRROCK1DGAT1JAK2JAK1
SCHEMBL790400 0.85 PI4KA (0.48) ATRPI4KAPIK3CGMAPTDGAT1
SCHEMBL789511 0.85 SMN1; SMN2 (0.59) ATRTP53SMN1; SMN2MAPTMAPK14
SCHEMBL790786 0.85 ALDH1A1 (0.52) PI4KAPIK3CGMAPTJAK2JAK1
SCHEMBL789721 0.81 MAPK14 (0.51) SMN1; SMN2MAPTMAPK14NPC1RAB9A
SCHEMBL791145 0.81 KDR (0.46) TP53MAPK1MAPTHDAC1NPC1
SCHEMBL789670 0.77 PI4KA (0.51) TP53SMN1; SMN2MAPK1PI4KAPIK3CG
SCHEMBL807273 0.76 ALDH1A1 (0.53) TP53SMN1; SMN2PI4KAPIK3CGJAK2
SCHEMBL789696 0.73 JAK2 (0.48) TP53SMN1; SMN2MAPK1PI4KAPIK3CG
Formic Acid SCHEMBL790534 0.73 ALDH1A1 (0.50) SMN1; SMN2PI4KAPIK3CGJAK2JAK1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2012037108-A1 AMINOQUINOLINE DERIVATIVES AS ANTIVIRAL AGENTS GLAXOSMITHKLINE LLC (US) 2012-03-22 WO disclosed
WO-2012037108-A1 AMINOQUINOLINE DERIVATIVES AS ANTIVIRAL AGENTS GLAXOSMITHKLINE LLC (US) 2012-03-22 WO disclosed