SCHEMBL790788

SCHEMBL790788

Nc1nc2ccc(-c3cccc(NC(=O)c4ccccc4)c3)cc2cc1-c1ccc(N2CCOCC2)cc1

nearest known ligand 0.54

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
NPC1 O15118 1/20 0.54
RAB9A P51151 1/20 0.54
MAPK14 Q16539 3/20 0.51
ATR Q13535 2/20 0.51
BTK Q06187 6/20 0.48
JAK2 O60674 1/20 0.48
JAK1 P23458 1/20 0.48
TYK2 P29597 1/20 0.48
JAK3 P52333 1/20 0.48
RPS6KA2 Q15349 1/20 0.47
SCN9A Q15858 1/20 0.47
EGFR P00533 1/20 0.47
ERBB2 P04626 1/20 0.47
IGF1R P08069 1/20 0.47
ROCK1 Q13464 1/20 0.47
DGAT1 O75907 1/20 0.46

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL789511 0.91 SMN1; SMN2 (0.59) NPC1RAB9AMAPK14ATR
SCHEMBL789721 0.91 MAPK14 (0.51) NPC1RAB9AMAPK14BTK
SCHEMBL790553 0.91 ATR (0.49) NPC1RAB9AMAPK14ATRJAK2
SCHEMBL807273 0.85 ALDH1A1 (0.53) NPC1RAB9AJAK2JAK1JAK3
SCHEMBL789670 0.83 PI4KA (0.51) NPC1RAB9A
Formic Acid SCHEMBL790534 0.82 ALDH1A1 (0.50) JAK2JAK1JAK3
SCHEMBL790535 0.80 PI4KA (0.41) MAPK14ATRBTKJAK2JAK1
SCHEMBL789915 0.80 RAB9A (0.50) NPC1RAB9ABTK
SCHEMBL789696 0.80 JAK2 (0.48) NPC1RAB9AJAK2
SCHEMBL790400 0.76 PI4KA (0.48) ATRJAK2DGAT1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2012037108-A1 AMINOQUINOLINE DERIVATIVES AS ANTIVIRAL AGENTS GLAXOSMITHKLINE LLC (US) 2012-03-22 WO disclosed
WO-2012037108-A1 AMINOQUINOLINE DERIVATIVES AS ANTIVIRAL AGENTS GLAXOSMITHKLINE LLC (US) 2012-03-22 WO disclosed