SCHEMBL7908313

SCHEMBL7908313

COc1ccc(N(C)c2ccc(C(=O)c3ccc(OC(F)F)c(OC(F)F)c3)cn2)cc1

nearest known ligand 0.44

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 1/20 0.44
GAA P10253 1/20 0.44
PDE4A P27815 4/20 0.42
PDE4B Q07343 4/20 0.41
PDE4C Q08493 3/20 0.41
PDE4D Q08499 3/20 0.41
RXFP1 Q9HBX9 1/20 0.41
LTC4S Q16873 2/20 0.39
TUBB4A P04350 1/20 0.38
TUBB P07437 1/20 0.38
TUBA3C P0DPH7 1/20 0.38
TUBA1B P68363 1/20 0.38
TUBA4A P68366 1/20 0.38
TUBB4B P68371 1/20 0.38
TUBB3 Q13509 1/20 0.38
TUBB2A Q13885 1/20 0.38
TUBB8 Q3ZCM7 1/20 0.38
TUBA3E Q6PEY2 1/20 0.38
TUBA1A Q71U36 1/20 0.38
TUBA1C Q9BQE3 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7906572 0.80 PDE4A (0.51) PDE4AHPGDCASP1MEN1KMT2A
SCHEMBL10392397 0.77 CYP1A2 (0.54) ALDH1A1GAAPDE4DHPGDCYP1A2
SCHEMBL4827006 0.74 ALDH1A1 (0.53) ALDH1A1GAAPDE4APDE4BPDE4C
SCHEMBL7904298 0.73 PDE4A (0.43) PDE4APDE4BPDE4CPDE4DHPGD
SCHEMBL7991282 0.72 LMNA (0.54) ALDH1A1GAAPDE4APDE4BPDE4C
SCHEMBL7908376 0.72 PDE4A (0.44) ALDH1A1PDE4APDE4BPDE4CPDE4D
SCHEMBL7905359 0.72 PDE4A (0.65) PDE4A
SCHEMBL17602246 0.71 MAPT (0.41) GAARXFP1LTC4STUBB4ATUBB
SCHEMBL27830996 0.69 LTC4S (0.41) LTC4SRXRAMAPT
SCHEMBL7994597 0.68 LMNA (0.43) PDE4APDE4BPDE4CPDE4DVNN1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6200993-B1 ASTHMA; ANTIINFLAMMATORY AGENTS MERCK FROSST CANADA & CO. (CA) 2001-03-13 US disclosed