SCHEMBL7908376

SCHEMBL7908376

O=C(c1ccc(Br)nc1)c1ccc(OC(F)F)c(OC(F)F)c1

nearest known ligand 0.44

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
PDE4A P27815 11/20 0.44
PDE4B Q07343 10/20 0.44
PDE4C Q08493 9/20 0.44
PDE4D Q08499 9/20 0.44
ABCB11 O95342 1/20 0.39
ALDH1A1 P00352 1/20 0.39
KDM4E B2RXH2 1/20 0.38
HTT P42858 1/20 0.38
CYP1A2 P05177 1/20 0.38
CYP3A4 P08684 1/20 0.38
CYP2C9 P11712 1/20 0.38
TSHR P16473 1/20 0.38
CYP2C19 P33261 1/20 0.38
L3MBTL1 Q9Y468 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5973043 0.76 RXFP1 (0.44) ALDH1A1HTTCYP1A2CYP2C9CYP2C19
SCHEMBL4160646 0.76 PDE4A (0.61) PDE4APDE4BPDE4CPDE4DALDH1A1
SCHEMBL7991282 0.74 LMNA (0.54) PDE4APDE4BPDE4CPDE4DALDH1A1
SCHEMBL7994597 0.74 LMNA (0.43) PDE4APDE4BPDE4CPDE4D
SCHEMBL7907874 0.74 PDE4A (0.53) PDE4APDE4BPDE4CPDE4D
SCHEMBL7367599 0.73 PDE4A (0.43) PDE4A
SCHEMBL7908313 0.72 ALDH1A1 (0.44) PDE4APDE4BPDE4CPDE4DALDH1A1
SCHEMBL7994711 0.72 RAB9A (0.49) PDE4APDE4BPDE4CPDE4DALDH1A1
SCHEMBL1029279 0.72 PDE4A (0.59) PDE4APDE4BPDE4CPDE4DALDH1A1
SCHEMBL4827006 0.71 ALDH1A1 (0.53) PDE4APDE4BPDE4CPDE4DALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6200993-B1 ASTHMA; ANTIINFLAMMATORY AGENTS MERCK FROSST CANADA & CO. (CA) 2001-03-13 US disclosed
US-6180650-B1 ANTIINFLAMMATORY AGENTS; RESPIRATORY SYSTEM DISORDERS; SKIN DISORDERS; ANTITUMOR AGENTS MERCK FROSST CANADA & CO. (CA) 2001-01-30 US disclosed