SCHEMBL7908424

SCHEMBL7908424

NC(=O)c1cccc(-c2ccc(N)c3ccccc23)c1F

nearest known ligand 0.43

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
BTK Q06187 1/20 0.43
KEAP1 Q14145 2/20 0.43
NFE2L2 Q16236 2/20 0.43
CRHBP P24387 1/20 0.43
CRHR2 Q13324 1/20 0.43
KDM4E B2RXH2 3/20 0.42
ALDH1A1 P00352 2/20 0.42
GAA P10253 1/20 0.42
BCAT2 O15382 1/20 0.42
ALOX5AP P20292 1/20 0.41
FEN1 P39748 1/20 0.41
PARP1 P09874 2/20 0.41
POLB P06746 2/20 0.40
SMN1; SMN2 Q16637 1/20 0.40
CDC25B P30305 1/20 0.40
NPC1 O15118 1/20 0.40
RAB9A P51151 1/20 0.40
NSD2 O96028 2/20 0.39
BRD4 O60885 1/20 0.39
PDK2 Q15119 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL17599359 0.88 CDC25B (0.50) KEAP1NFE2L2CRHBPCRHR2KDM4E
SCHEMBL30881836 0.77 KEAP1 (0.44) BTKKEAP1BCAT2ALOX5APFEN1
SCHEMBL30646218 0.75 BCAT2 (0.63) BTKKEAP1NFE2L2KDM4EALDH1A1
SCHEMBL30841448 0.75 BCAT2 (0.69) KEAP1NFE2L2CRHBPCRHR2KDM4E
SCHEMBL27651120 0.74 MMP2 (0.45) BTKKEAP1NFE2L2KDM4EALDH1A1
SCHEMBL6061358 0.74 ALDH1A1 (0.56) KEAP1KDM4EALDH1A1GAAPARP1
SCHEMBL5748491 0.74 ATM (0.62) BTKKDM4EALDH1A1GAABCAT2
SCHEMBL30623038 0.74 MMP2 (0.45) BTKKEAP1NFE2L2KDM4EALDH1A1
SCHEMBL634722 0.73 ATM (0.55) KEAP1NFE2L2KDM4EALDH1A1GAA
SCHEMBL29733181 0.73 PARP1 (0.58) KEAP1NFE2L2ALDH1A1GAABCAT2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6197803-B1 VIRICIDES; PREVENTION REPRODUCTION AMERICAN HOME PRODUCTS CORPORATION 2001-03-06 US disclosed