SCHEMBL790895

SCHEMBL790895

COc1ncc(Br)cc1NS(=O)(=O)c1cccc2cccnc12

nearest known ligand 0.61

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 3/20 0.61
POLB P06746 1/20 0.61
TSHR P16473 1/20 0.60
MEN1 O00255 7/20 0.59
KMT2A Q03164 7/20 0.59
TP53 P04637 1/20 0.57
HTT P42858 1/20 0.57
ATM Q13315 1/20 0.56
SLC40A1 Q9NP59 4/20 0.56
GAA P10253 1/20 0.53
MAPT P10636 2/20 0.52
HPGD P15428 1/20 0.52
NPSR1 Q6W5P4 1/20 0.52

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL29255664 0.81 MEN1 (0.62) ALDH1A1POLBMEN1KMT2AATM
SCHEMBL30854812 0.81 MEN1 (0.62) ALDH1A1POLBMEN1KMT2AATM
SCHEMBL791091 0.80 ALPL (0.57) ALDH1A1POLBTSHRMEN1KMT2A
SCHEMBL30902213 0.79 PIK3CA (0.56) TSHR
SCHEMBL15555632 0.79 PIK3CA (0.56) TSHR
SCHEMBL790388 0.79 PIK3CG (0.56) ALDH1A1POLBTSHRMEN1KMT2A
SCHEMBL789565 0.78 PIK3CA (0.57) SLC40A1GAA
SCHEMBL791058 0.78 GLO1 (0.47) SLC40A1
SCHEMBL29255671 0.77 CXCR2 (0.77) ALDH1A1POLBTSHRMEN1KMT2A
SCHEMBL30854819 0.77 CXCR2 (0.77) ALDH1A1POLBTSHRMEN1KMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2012087938-A1 QUINAZOLINONE DERIVATIVES AS ANTIVIRAL AGENTS GLAXOSMITHKLINE LLC (US) 2012-06-28 WO disclosed
WO-2012087938-A1 QUINAZOLINONE DERIVATIVES AS ANTIVIRAL AGENTS GLAXOSMITHKLINE LLC (US) 2012-06-28 WO disclosed
WO-2012037108-A1 AMINOQUINOLINE DERIVATIVES AS ANTIVIRAL AGENTS GLAXOSMITHKLINE LLC (US) 2012-03-22 WO disclosed
WO-2012037108-A1 AMINOQUINOLINE DERIVATIVES AS ANTIVIRAL AGENTS GLAXOSMITHKLINE LLC (US) 2012-03-22 WO disclosed