SCHEMBL7909434

SCHEMBL7909434

COC(=O)CCN1CCN(C(=O)CN2CCN(C(=N)N)CC2)CC1

nearest known ligand 0.50

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
SMN1; SMN2 Q16637 2/20 0.50
PKM P14618 1/20 0.47
GAA P10253 1/20 0.40
GLA P06280 1/20 0.38
ALOX15 P16050 1/20 0.38
TSHR P16473 1/20 0.38
HSD17B10 Q99714 1/20 0.38
KMT2A Q03164 3/20 0.37
MEN1 O00255 1/20 0.36
KDM1A O60341 1/20 0.36
DRD3 P35462 1/20 0.36
ALDH1A1 P00352 4/20 0.36
MAPT P10636 2/20 0.36
TPSAB1 Q15661 2/20 0.36
TPSD1 Q9BZJ3 2/20 0.36
TPSG1 Q9NRR2 2/20 0.36
HTT P42858 1/20 0.36
KDM4E B2RXH2 1/20 0.36
LMNA P02545 1/20 0.35
CACNA1C Q13936 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8380855 0.92 PKM (0.45) SMN1; SMN2PKMGAAGLAALOX15
SCHEMBL8382459 0.88 PKM (0.51) SMN1; SMN2PKMGAAGLAALOX15
SCHEMBL7909740 0.84 SMN1; SMN2 (0.46) SMN1; SMN2PKMGLAKMT2AMEN1
SCHEMBL8384455 0.82 PKM (0.45) PKMGAAGLAALOX15TSHR
SCHEMBL19146051 0.82 PKM (0.42) SMN1; SMN2PKMTSHRKMT2AKDM1A
SCHEMBL8384378 0.77 MAPK1 (0.47) SMN1; SMN2PKMGAAALOX15TSHR
SCHEMBL4489670 0.76 SMN1; SMN2 (0.65) SMN1; SMN2GLATSHRKMT2AMEN1
SCHEMBL1174392 0.76
SCHEMBL8381872 0.76 PKM (0.40) SMN1; SMN2PKMTSHRKMT2AKDM1A
SCHEMBL7913433 0.76 GAA (0.50) PKMGAAALOX15TSHRHSD17B10

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0608759-B1 Piperazine derivatives MERCK PATENT GMBH (DE) 2001-08-22 EP disclosed
US-5908843-A Piperazine compounds as fibrinogen inhibitors MERCK PATENT GESELLSCHAFT MIT BESCHRANKTER HAFTUNG (DE) 1999-06-01 US disclosed
EP-0608759-A2 Piperazinderivatives MERCK PATENT GmbH (DE) 1994-08-03 EP disclosed