SCHEMBL7913433

SCHEMBL7913433

N=C(N)N1CCN(CC(=O)N2CCN(CC(=O)O)CC2)CC1

nearest known ligand 0.54

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
GAA P10253 1/20 0.50
PKM P14618 2/20 0.49
HSD17B10 Q99714 2/20 0.47
ALOX15 P16050 1/20 0.47
TSHR P16473 1/20 0.47
ALDH1A1 P00352 4/20 0.46
MAPT P10636 2/20 0.46
MAPK1 P28482 1/20 0.42
CPN1 P15169 1/20 0.38
CPB2 Q96IY4 1/20 0.38
TPSAB1 Q15661 2/20 0.38
TPSD1 Q9BZJ3 2/20 0.38
TPSG1 Q9NRR2 2/20 0.38
F2 P00734 1/20 0.38
NPSR1 Q6W5P4 1/20 0.38
KDM4E B2RXH2 1/20 0.37
TDP1 Q9NUW8 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7900115 0.93 MAPK1 (0.46) GAAPKMHSD17B10ALOX15TSHR
SCHEMBL8384455 0.87 PKM (0.45) GAAPKMHSD17B10ALOX15TSHR
SCHEMBL7127595 0.87 GAA (0.64) GAAPKMHSD17B10ALOX15TSHR
SCHEMBL8384378 0.84 MAPK1 (0.47) GAAPKMHSD17B10ALOX15TSHR
SCHEMBL8386026 0.83 ITGB3 (0.40) GAAPKMHSD17B10TSHRALDH1A1
SCHEMBL7129737 0.81 GAA (0.63) GAAHSD17B10ALOX15TSHRALDH1A1
SCHEMBL8382459 0.80 PKM (0.51) GAAPKMHSD17B10ALOX15TSHR
SCHEMBL5872643 0.79 GAA (0.65) GAAHSD17B10ALOX15TSHRALDH1A1
SCHEMBL19146559 0.79 KDM4E (0.52) GAAPKMHSD17B10ALOX15TSHR
SCHEMBL15499763 0.77 BLM (0.49) GAAPKMHSD17B10ALOX15TSHR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0608759-B1 Piperazine derivatives MERCK PATENT GMBH (DE) 2001-08-22 EP disclosed
US-5908843-A Piperazine compounds as fibrinogen inhibitors MERCK PATENT GESELLSCHAFT MIT BESCHRANKTER HAFTUNG (DE) 1999-06-01 US disclosed
EP-0608759-A2 Piperazinderivatives MERCK PATENT GmbH (DE) 1994-08-03 EP disclosed