SCHEMBL7920801

SCHEMBL7920801

COc1cccc2c1OC(CO)CN2C(=O)OC(C)(C)C

nearest known ligand 0.42

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KDM4E B2RXH2 1/20 0.42
ALDH1A1 P00352 1/20 0.42
HPGD P15428 1/20 0.42
PRKCA P17252 1/20 0.38
DRD2 P14416 4/20 0.38
NOTUM Q6P988 1/20 0.38
RORC P51449 4/20 0.37
TP53 P04637 2/20 0.37
MAPT P10636 1/20 0.37
PDE4B Q07343 1/20 0.37
KDM1A O60341 1/20 0.36
HDAC1 Q13547 1/20 0.36
HDAC6 Q9UBN7 1/20 0.36
CACNB4 O00305 1/20 0.36
CACNA1A O00555 1/20 0.36
CACNA1G O43497 1/20 0.36
CACNG3 O60359 1/20 0.36
CACNA1F O60840 1/20 0.36
CACNA1H O95180 1/20 0.36
CACNB3 P54284 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3205346 0.88 UCHL1 (0.44) RORCKDM1AHDAC1HDAC6
SCHEMBL30479646 0.88 UCHL1 (0.44) RORCKDM1AHDAC1HDAC6
SCHEMBL7911444 0.82 ALDH1A1 (0.38) ALDH1A1HPGDRORCMAPTHTR1A
SCHEMBL6975852 0.81 RORC (0.45) RORCTP53MAPTKDM1AMEN1
SCHEMBL7919024 0.77 KDM4E (0.46) KDM4EALDH1A1HPGDPRKCADRD2
SCHEMBL6977474 0.76 MAPT (0.44) ALDH1A1RORCTP53MAPT
SCHEMBL7918936 0.75 HTR1A (0.47) KDM4EALDH1A1HPGDPRKCATP53
SCHEMBL22396991 0.74 RORC (0.52) RORCTP53MAPT
SCHEMBL22396988 0.74 RORC (0.52) RORCTP53MAPT
SCHEMBL22397004 0.74 RORC (0.52) RORCTP53MAPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6221863-B1 TREATING DEPRESSION IN A PATIENT AMERICAN HOME PRODUCTS CORP. 2001-04-24 US disclosed
WO-2000040581-A1 3,4-DIHYDRO-2H-BENZO[1,4]OXAZINE DERIVATIVES AMERICAN HOME PRODUCTS CORPORATION (US) 2000-07-13 WO disclosed