SCHEMBL7920931

SCHEMBL7920931

COc1cc(C(O)CNC(=O)c2ccc3c(c2)c(Cl)cn3C)cc(OC)c1OC

nearest known ligand 0.43

Predicted protein targets (top 10)

geneUniProtsupporting neighboursconfidence
TP53 P04637 2/20 0.42
HDAC11 Q96DB2 1/20 0.42
HDAC8 Q9BY41 1/20 0.42
HDAC6 Q9UBN7 1/20 0.42
MAPT P10636 1/20 0.42
CPT1A P50416 2/20 0.42
CPT2 P23786 1/20 0.42
CPT1B Q92523 1/20 0.42
ROCK2 O75116 5/20 0.41
ROCK1 Q13464 5/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7930108 0.79 KMT2A (0.57) TP53ROCK2ROCK1
SCHEMBL7927749 0.78 ALDH1A1 (0.57) MAPTROCK2ROCK1
SCHEMBL7930156 0.73 HPGD (0.57) HDAC8HDAC6MAPT
SCHEMBL7929603 0.72 SMYD3 (0.45) TP53MAPTROCK2ROCK1
SCHEMBL7928025 0.70 SMPD1 (0.56) HDAC8HDAC6MAPTROCK2ROCK1
SCHEMBL7927928 0.68 TP53 (0.49) TP53MAPT
SCHEMBL7929624 0.67 NR4A2 (0.44) TP53MAPTROCK2ROCK1
SCHEMBL8910176 0.66 TDP1 (0.53) TP53MAPTROCK2ROCK1
SCHEMBL11818791 0.65 KMT2A (0.52) TP53
SCHEMBL19125501 0.64 HDAC6 (0.68) HDAC11HDAC8HDAC6

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6228868-B1 ANTICARCINOGENIC AND ANTITUMOR AGENTS ABBOTT LABORATORIES 2001-05-08 US disclosed