SCHEMBL7932797

SCHEMBL7932797

O=C(CS)Nc1ccc(Cl)c(Cl)c1

nearest known ligand 1.00 ✓ in ChEMBL — recovers established targets

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CYP3A4 P08684 1/20 0.69
EPHX1 P07099 2/20 0.63
EPHX2 P34913 2/20 0.63
MAPT P10636 4/20 0.59
NPSR1 Q6W5P4 2/20 0.59
ALDH1A1 P00352 1/20 0.59
ALOX15 P16050 1/20 0.59
HSD17B10 Q99714 1/20 0.59
MEN1 O00255 4/20 0.59
KMT2A Q03164 4/20 0.59
L3MBTL1 Q9Y468 2/20 0.59
POLB P06746 1/20 0.59
NPC1 O15118 3/20 0.58
LMNA P02545 2/20 0.58
HTT P42858 2/20 0.58
RAB9A P51151 2/20 0.58
HSP90AA1 P07900 1/20 0.58
NPY1R P25929 1/20 0.58
NPY2R P49146 1/20 0.58
SMN1; SMN2 Q16637 1/20 0.58

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL23857903 0.86 CYP3A4 (0.65) CYP3A4EPHX1EPHX2MAPTNPSR1
SCHEMBL7933287 0.84 TSHR (0.71) MAPTNPSR1ALDH1A1MEN1KMT2A
SCHEMBL7929903 0.84 NPC1 (0.59) CYP3A4MAPTALDH1A1ALOX15MEN1
SCHEMBL7923953 0.84 MAPT (0.54) CYP3A4EPHX1EPHX2MAPTNPSR1
SCHEMBL4003878 0.83 CYP3A4 (0.71) CYP3A4EPHX1EPHX2MAPTNPSR1
SCHEMBL30833308 0.83 CYP3A4 (0.71) CYP3A4EPHX1EPHX2MAPTNPSR1
Propanil SCHEMBL26871 0.81 CYP3A4 (1.00) CYP3A4EPHX1EPHX2MAPTNPSR1
Propanil SCHEMBL1702271 0.81 CYP3A4 (1.00) CYP3A4EPHX1EPHX2MAPTNPSR1
Propanil SCHEMBL21900164 0.81 CYP3A4 (1.00) CYP3A4EPHX1EPHX2MAPTNPSR1
SCHEMBL15107476 0.81 L3MBTL1 (0.74) CYP3A4EPHX1EPHX2MAPTNPSR1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20110190285-A1 METHODS OF TREATING A BOTULINUM TOXIN RELATED CONDITION IN A SUBJECT ABSOLUTE SCIENCE, INC. (US) 2011-08-04 US disclosed
US-20110034521-A1 COMPOUNDS AND METHODS FOR TREATING ZINC MATRIX METALLOPROTEASE DEPENDENT DISEASES NATIONAL INSTITUTES OF HEALTH (NIH), U.S. DEPT. OF HEALTH AND HUMAN SERVICES (DHHS), U.S. GOVERNMENT 2011-02-10 US disclosed
WO-2010033360-A1 METHODS OF TREATING A BOTULINUM TOXIN RELATED CONDITION IN A SUBJECT 1/3 ABSOLUTE SCIENCE, INC. (US) 2010-03-25 WO disclosed
WO-2009045761-A1 COMPOUNDS AND METHODS FOR TREATING ZINC MATRIX METALLOPROTEASE DEPENDENT DISEASES ABSOLUTE SCIENCE, INC. (US) 2009-04-09 WO disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (2 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20110034521-A1 COMPOUNDS AND METHODS FOR TREATING ZINC MATRIX METALLOPROTEASE DEPENDENT DISEASES MMP7, MMP3, MMP9 CYP3A4 3370/4885EPHX1 565/4885EPHX2 1173/4885
US-20110190285-A1 METHODS OF TREATING A BOTULINUM TOXIN RELATED CONDITION IN A SUBJECT NPY5R, RAC3, CPA3 CYP3A4 2145/4885EPHX1 1273/4885EPHX2 940/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.