SCHEMBL7937185

SCHEMBL7937185

COC(=O)C(Sc1ccc2c(c1)OCO2)C(C)(c1ccccc1)c1ccccc1

nearest known ligand 0.44

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
EDNRA P25101 5/20 0.44
ALDH1A1 P00352 2/20 0.44
TSHR P16473 2/20 0.44
LMNA P02545 1/20 0.44
KIF11 P52732 1/20 0.41
MEN1 O00255 1/20 0.41
KMT2A Q03164 1/20 0.41
POLB P06746 2/20 0.40
NPC1 O15118 4/20 0.40
RAB9A P51151 4/20 0.40
MAPT P10636 2/20 0.40
SMN1; SMN2 Q16637 2/20 0.40
NFKB1 P19838 1/20 0.40
NFKB2 Q00653 1/20 0.40
RELA Q04206 1/20 0.40
CYP1A2 P05177 1/20 0.40
CYP3A4 P08684 1/20 0.40
CYP2D6 P10635 1/20 0.40
CYP2C9 P11712 1/20 0.40
MAPK1 P28482 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8091800 0.88 KIF11 (0.46) EDNRAALDH1A1TSHRLMNAKIF11
SCHEMBL7936594 0.75 KMT2A (0.45) ALDH1A1TSHRLMNAMEN1KMT2A
SCHEMBL7937232 0.72 KDM4E (0.44) EDNRAALDH1A1LMNAMEN1KMT2A
SCHEMBL7937196 0.69 EDNRB (0.49) EDNRA
SCHEMBL7394832 0.68 SMN1; SMN2 (0.48) EDNRAALDH1A1TSHRNPC1RAB9A
SCHEMBL16697795 0.67 RAB9A (0.47) ALDH1A1MEN1KMT2ANPC1RAB9A
SCHEMBL16697151 0.67 RAB9A (0.47) ALDH1A1MEN1KMT2ANPC1RAB9A
SCHEMBL1746047 0.67 PTGS2 (0.56) EDNRAALDH1A1MEN1KMT2ATAS1R3
SCHEMBL9459877 0.66 GSTP1 (0.47) ALDH1A1TSHRLMNANPC1RAB9A
SCHEMBL7934306 0.66 EDNRB (0.46) EDNRAALDH1A1TSHRLMNAMEN1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6235903-B1 Method for preparing sulfanyl-type endothelin receptor antagonists BASF AKTIENGESELLSCHAFT (DE) 2001-05-22 US disclosed