SCHEMBL7937531

SCHEMBL7937531

COc1ccc(C#CCS(=O)(=O)c2ccc(C)cc2)cc1

nearest known ligand 0.51

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 7/20 0.51
GAA P10253 1/20 0.51
MAPT P10636 2/20 0.49
CYP1A2 P05177 1/20 0.49
CYP3A4 P08684 1/20 0.49
CYP2C9 P11712 1/20 0.49
CYP2C19 P33261 1/20 0.49
HPGD P15428 1/20 0.48
KMT2A Q03164 1/20 0.48
TDP1 Q9NUW8 1/20 0.48
ACHE P22303 2/20 0.47
BCHE P06276 1/20 0.47
CA12 O43570 1/20 0.45
CA1 P00915 1/20 0.45
CA2 P00918 1/20 0.45
CA9 Q16790 1/20 0.45
MMP13 P45452 2/20 0.44
MMP8 P22894 1/20 0.44
MMP2 P08253 1/20 0.44
MMP3 P08254 1/20 0.44

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL28641212 0.80 ALDH1A1 (0.62) ALDH1A1GAAMAPTKMT2AMMP13
SCHEMBL7924997 0.79 LMNA (0.52) ALDH1A1MAPTCYP3A4CYP2C9CYP2C19
SCHEMBL29118794 0.79 APP (0.48) ALDH1A1MAPTCYP1A2CYP3A4CYP2C9
SCHEMBL7931631 0.78 ALDH1A1 (0.59) ALDH1A1GAAMAPTCYP1A2CYP3A4
SCHEMBL28440362 0.77 CA12 (0.49) ALDH1A1GAAHPGDKMT2AACHE
SCHEMBL10825960 0.77 ALDH1A1 (0.59) ALDH1A1GAAMAPTCYP1A2CYP3A4
SCHEMBL6424729 0.76 MMP13 (0.50) ALDH1A1GAAKMT2ACA12CA1
SCHEMBL10525794 0.75 ACHE (0.71) ALDH1A1GAAMAPTHPGDKMT2A
SCHEMBL10420685 0.74 MMP13 (0.58) ALDH1A1GAAMAPTKMT2AMMP13
SCHEMBL7935192 0.73 PKM (0.57) ALDH1A1GAAMAPTCYP1A2CYP3A4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6242478-B1 ANTICARCINOGENIC AGENTS; REPLICATION INHIBITORS OF HUMAN LYMPHADENOPATHY ASSOCIATED VIRUS(HIV) WAKE FOREST UNIVERSITY 2001-06-05 US disclosed