SCHEMBL7937864

SCHEMBL7937864

CCn1c(=O)c(-c2nccs2)nc2c(N)cc(NCc3c(F)cccc3F)nc21

nearest known ligand 0.38

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ADORA2A P29274 7/20 0.38
ADORA1 P30542 7/20 0.38
ADORA2B P29275 3/20 0.38
ADORA3 P0DMS8 2/20 0.36
LYN P07948 1/20 0.35
PDE4B Q07343 2/20 0.35
PDE7A Q13946 1/20 0.35
USP2 O75604 2/20 0.33
ALDH1A1 P00352 2/20 0.33
CYP1A2 P05177 2/20 0.33
CYP3A4 P08684 2/20 0.33
CASP1 P29466 2/20 0.33
CASP7 P55210 2/20 0.33
HIF1A Q16665 2/20 0.33
HSD17B10 Q99714 2/20 0.33
HPGD P15428 1/20 0.33
PDE4A P27815 1/20 0.33
PDE4C Q08493 1/20 0.33
PDE4D Q08499 1/20 0.33
PDE3B Q13370 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7937752 0.93 ADORA2A (0.39) ADORA2AADORA1ADORA2BADORA3LYN
SCHEMBL7943995 0.78 HSF1 (0.36) ADORA2AADORA1ADORA3LYNPDE7A
SCHEMBL7937747 0.77 HSF1 (0.35) ADORA2AADORA1ADORA3LYNPDE7A
SCHEMBL7946794 0.76 ADORA1 (0.39) ADORA2AADORA1ADORA2BADORA3LYN
SCHEMBL7944574 0.75 HSF1 (0.36) ADORA2AADORA1ADORA2BADORA3LYN
SCHEMBL7943760 0.74 CD38 (0.37) ADORA2AADORA1ADORA2BUSP2ALDH1A1
SCHEMBL7944093 0.72 STIM1 (0.38) ADORA2AADORA1ADORA2BALDH1A1CYP3A4
SCHEMBL7945987 0.68 TYRO3 (0.36) USP2ALDH1A1CYP1A2CASP1CASP7
SCHEMBL7944078 0.67 PDE4B (0.42) ADORA2AADORA1ADORA2BADORA3PDE4B
SCHEMBL7947006 0.67 ALDH1A1 (0.34) ADORA2AADORA1ADORA2BLYNUSP2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2010008775-A1 AMINOPYRIDOPYRAZINONE DERIVATIVES FOR TREATING NEURODEGENERATIVE DISEASES LIGAND PHARMACEUTICALS INC. (US) 2010-01-21 WO disclosed