SCHEMBL7938599

SCHEMBL7938599

FC(F)(c1ccccc1)c1ccc(Cl)cc1

nearest known ligand 0.48

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
TSHR P16473 4/20 0.48
ALDH1A1 P00352 1/20 0.48
CYP19A1 P11511 4/20 0.47
KIF11 P52732 3/20 0.47
CYP1A2 P05177 1/20 0.46
L3MBTL1 Q9Y468 3/20 0.44
HTT P42858 2/20 0.44
SMN1; SMN2 Q16637 2/20 0.44
CNR1 P21554 1/20 0.41
MEN1 O00255 2/20 0.41
KMT2A Q03164 2/20 0.41
MAPK1 P28482 2/20 0.41
HIF1A Q16665 1/20 0.41
BCL2 P10415 1/20 0.41
LMNA P02545 1/20 0.40
CYP2A6 P11509 1/20 0.40
XBP1 P17861 1/20 0.40
NPSR1 Q6W5P4 1/20 0.40
MIF P14174 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL809832 0.89 LMNA (0.50) TSHRCYP19A1MEN1KMT2AMAPK1
SCHEMBL1108511 0.84 TSHR (0.65) TSHRALDH1A1KIF11CYP1A2MAPK1
SCHEMBL28021962 0.81 TSHR (0.61) TSHRALDH1A1KIF11CYP1A2MAPK1
SCHEMBL3949150 0.79 TSHR (0.53) TSHRCYP19A1KIF11CYP1A2L3MBTL1
SCHEMBL8157070 0.79 TSHR (0.53) TSHRCYP19A1KIF11CYP1A2L3MBTL1
SCHEMBL9263367 0.78 CA1 (0.42) TSHRCYP19A1HTTSMN1; SMN2MEN1
SCHEMBL367665 0.77 CYP19A1 (0.61) TSHRCYP19A1KIF11CYP1A2L3MBTL1
SCHEMBL2864477 0.77 TSHR (0.61) TSHRCYP19A1KIF11CYP1A2L3MBTL1
SCHEMBL11652133 0.77 CYP19A1 (0.61) TSHRCYP19A1KIF11CYP1A2L3MBTL1
SCHEMBL11511851 0.77 TSHR (0.61) TSHRCYP19A1KIF11CYP1A2L3MBTL1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0730566-B1 SELECTIVELY FLUORINATED ORGANIC COMPOUNDS F2 CHEMICALS LTD (GB) 2001-09-19 EP disclosed
US-5789580-A Selectively fluorinated organic compounds BRITISH NUCLEAR FUELS PLC (GB) 1998-08-04 US disclosed
EP-0730566-A1 SELECTIVELY FLUORINATED ORGANIC COMPOUNDS BNFL FLUOROCHEMICALS LTD. (GB) 1996-09-11 EP disclosed
WO-1996003357-A1 SELECTIVELY FLUORINATED ORGANIC COMPOUNDS BNFL FLUOROCHEMICALS LTD. (GB) 1996-02-08 WO disclosed