SCHEMBL7946705

SCHEMBL7946705

CC(C)C[C@@H](C(=O)NN1C(=O)CNC1=O)[C@H](Cc1ccccc1-c1ccccc1)C(=O)NOC1CCCCO1

nearest known ligand 0.34

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ITGB1 P05556 2/20 0.34
ITGA4 P13612 2/20 0.34
SLC6A2 P23975 1/20 0.32
SLC6A4 P31645 1/20 0.32
XIAP P98170 1/20 0.32
CASP1 P29466 1/20 0.31
CASP3 P42574 1/20 0.31
CASP7 P55210 1/20 0.31
CASP6 P55212 1/20 0.31
CASP8 Q14790 1/20 0.31
NOTCH1 P46531 1/20 0.30
PSEN1 P49768 1/20 0.30
PSEN2 P49810 1/20 0.30
RBPJ Q06330 1/20 0.30
APH1B Q8WW43 1/20 0.30
NCSTN Q92542 1/20 0.30
APH1A Q96BI3 1/20 0.30
PSENEN Q9NZ42 1/20 0.30
MME P08473 1/20 0.30
ACE P12821 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7955767 0.89 ITGB1 (0.36) ITGB1ITGA4MMEACECPA1
SCHEMBL7828157 0.83 ADAM17 (0.39) CASP1CASP3CASP7CASP6CASP8
SCHEMBL7946622 0.82 MMP2 (0.41)
SCHEMBL7946619 0.82 MMP2 (0.41)
SCHEMBL7835182 0.82 MMP2 (0.41)
SCHEMBL6220706 0.79 BMP1 (0.33)
SCHEMBL6221034 0.77 MMP1 (0.38) PSEN1PSEN2APH1BNCSTNAPH1A
SCHEMBL7955118 0.77 MMP1 (0.37) PSEN1PSEN2APH1BNCSTNAPH1A
SCHEMBL6946530 0.74 ADAM17 (0.40) CASP1CASP3CASP7CASP6CASP8
SCHEMBL6946529 0.74 ADAM17 (0.40) CASP1CASP3CASP7CASP6CASP8

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6281363-B1 ANTIINFLAMMATORY AGENTS; ANTIARTHRITIC AGENTS; AUTOIMMUNE DISORDERS HOFFMANN-LA ROCHE INC. 2001-08-28 US disclosed