SCHEMBL7947475

SCHEMBL7947475

O=C(NCc1ccccc1N1CCN(c2ccncc2)CC1)c1ccccc1

nearest known ligand 0.57

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
KMT2A Q03164 1/20 0.52
PLA2G1B P04054 1/20 0.51
SMN1; SMN2 Q16637 1/20 0.51
ATG4B Q9Y4P1 1/20 0.51
SCN2A Q99250 2/20 0.50
SCN10A Q9Y5Y9 2/20 0.50
DRD2 P14416 1/20 0.48
DRD4 P21917 1/20 0.48
DRD3 P35462 1/20 0.48
HTR1A P08908 1/20 0.47
ADRA1A P35348 1/20 0.47
ALDH1A1 P00352 1/20 0.47
HPGD P15428 1/20 0.47

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7967171 0.91 KMT2A (0.54) KMT2ASCN2ASCN10ADRD2DRD4
SCHEMBL5334419 0.80 ALDH1A1 (0.51) KMT2ASCN2ASCN10ADRD2DRD4
SCHEMBL7947618 0.78 KMT2A (0.49) KMT2ADRD2HTR1A
Hydrochloric Acid SCHEMBL27908881 0.77 DRD2 (0.72) DRD2
SCHEMBL2355678 0.76 DRD3 (0.72) DRD2DRD4DRD3HTR1A
SCHEMBL7956445 0.75 NAMPT (0.52) DRD2HTR1A
SCHEMBL7956809 0.75 SETDB1 (0.53) KMT2ASMN1; SMN2HTR1AALDH1A1
SCHEMBL8635355 0.75 GAA (0.55) KMT2ASMN1; SMN2DRD2DRD3HTR1A
SCHEMBL5160692 0.74 HTR1A (0.59) HTR1AADRA1A
SCHEMBL13212055 0.73 POLB (0.62) KMT2ASCN2ASCN10ADRD2DRD4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6313127-B1 FOR THERAPY OF HYPERCHOLESTEROLEMIA OR ATHEROSCLEROSIS ZENECA LIMITED (GB) 2001-11-06 US disclosed
EP-0880501-A1 HETEROCYCLIC COMPOUNDS USEFUL AS PHARMACEUTICAL AGENTS ZENECA LIMITED (GB) 1998-12-02 EP disclosed
WO-1997028128-A1 HETEROCYCLIC COMPOUNDS USEFUL AS PHARMACEUTICAL AGENTS ZENECA LIMITED (GB) 1997-08-07 WO disclosed