SCHEMBL7958463

SCHEMBL7958463

CC(C)n1c(=O)[nH]c2nc[nH]c2c1=S

nearest known ligand 0.55

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ADORA2B P29275 8/20 0.51
ADORA2A P29274 4/20 0.51
PDE4A P27815 3/20 0.48
PDE4B Q07343 3/20 0.48
PDE4C Q08493 3/20 0.48
PDE4D Q08499 3/20 0.48
ADORA3 P0DMS8 7/20 0.46
TDP1 Q9NUW8 2/20 0.41
ACHE P22303 1/20 0.41
GDA Q9Y2T3 1/20 0.41
ALDH1A1 P00352 3/20 0.41
TP53 P04637 2/20 0.41
HPGD P15428 2/20 0.41
PTGS1 P23219 2/20 0.41
HBB P68871 2/20 0.41
SMN1; SMN2 Q16637 2/20 0.41
KDM4E B2RXH2 2/20 0.41
USP2 O75604 1/20 0.38
MAPK3 P27361 1/20 0.38
XDH P47989 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL12413533 0.84 ADORA2B (0.63) ADORA2BADORA2APDE4APDE4BPDE4C
SCHEMBL150602 0.75 ADORA2B (0.59) ADORA2BADORA2APDE4APDE4BPDE4C
SCHEMBL9845197 0.73 PDE4A (0.74) ADORA2BADORA2APDE4APDE4BPDE4C
SCHEMBL2917584 0.72 ADORA2B (0.55) ADORA2BADORA2APDE4APDE4BPDE4C
SCHEMBL897035 0.72 ADORA2B (0.55) ADORA2BADORA2APDE4APDE4BPDE4C
SCHEMBL20653044 0.71 ADORA2A (0.58) ADORA2BADORA2APDE4APDE4BPDE4C
SCHEMBL10535015 0.71 ADORA2A (0.57) ADORA2BADORA2APDE4APDE4BPDE4C
SCHEMBL9845195 0.71 ADORA2A (0.75) ADORA2BADORA2APDE4APDE4BPDE4C
SCHEMBL7035609 0.70 ADORA2B (0.52) ADORA2BADORA2APDE4APDE4BPDE4C
1-Methylxanthine SCHEMBL10996 0.68 ADORA2B (1.00) ADORA2BADORA2APDE4APDE4BPDE4C

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6268373-B1 ENZYME INHIBITORS EURO-CELTIQUE S.A. (LU) 2001-07-31 US disclosed