SCHEMBL7958545

SCHEMBL7958545

COc1ccc2c(c1)NC(OC(=O)C(=O)OC1CC(CN(C)C)Cc3ccc(OC)cc3N1)CC(CN(C)C)C2

nearest known ligand 0.43

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
METAP1 P53582 3/20 0.43
MCHR1 Q99705 3/20 0.42
CA1 P00915 2/20 0.36
CA2 P00918 2/20 0.36
ACHE P22303 2/20 0.36
MTNR1A P48039 2/20 0.35
CYP19A1 P11511 1/20 0.34
CYP26A1 O43174 1/20 0.34
SLC6A2 P23975 1/20 0.34
SLC6A4 P31645 1/20 0.34
SLC6A3 Q01959 1/20 0.34
HTR5A P47898 1/20 0.34
HTR2A P28223 1/20 0.34
HTR2C P28335 1/20 0.34
HRH1 P35367 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Oxalic Acid SCHEMBL7958543 0.75 MCHR1 (0.46) METAP1MCHR1CA1CA2ACHE
Hydrochloric Acid SCHEMBL4623245 0.74 METAP1 (0.49) METAP1MCHR1CYP19A1CYP26A1SLC6A2
SCHEMBL3247442 0.70 ALOX15 (0.40) MTNR1A
SCHEMBL13937919 0.68 HTR5A (0.44) ACHECYP19A1HTR5AHTR2AHTR2C
SCHEMBL3241271 0.67 GAA (0.57) CA1CA2ACHEMTNR1AHTR5A
Hydrochloric Acid SCHEMBL4623292 0.66 CYP19A1 (0.59) METAP1MCHR1CA1CA2ACHE
Hydrochloric Acid SCHEMBL4622581 0.66 MCHR1 (0.59) METAP1MCHR1CA1CA2ACHE
SCHEMBL28634734 0.66 MTNR1A (0.44) CA1CA2ACHEMTNR1AHTR5A
SCHEMBL4999513 0.66 MTNR1A (0.44) CA1CA2ACHEMTNR1AHTR5A
SCHEMBL1321069 0.64 ALOX15 (0.44)

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6329389-B1 HETEROCYCLIC AMINES AND DERIVATIVES, SOMATOSTATIN AND ANTIDIABETIC AGENTS TAKEDA CHEMICAL INDUSTRIES, LTD. (JP) 2001-12-11 US disclosed