SCHEMBL796114

SCHEMBL796114

Cc1ccc(S(=O)(=O)NC(CCCCN)C(=O)O)cc1.O=CCCl

nearest known ligand 0.65

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MMP9 P14780 10/20 0.65
MMP2 P08253 9/20 0.65
ITGB3 P05106 1/20 0.50
ITGA2B P08514 1/20 0.50
TDP1 Q9NUW8 1/20 0.49
SLC1A3 P43003 1/20 0.46
SLC1A2 P43004 1/20 0.46
SLC1A1 P43005 1/20 0.46
MMP13 P45452 3/20 0.46
MMP3 P08254 2/20 0.46
L3MBTL1 Q9Y468 1/20 0.45
MMP8 P22894 1/20 0.44
ADAMTS4 O75173 1/20 0.44
PLAU P00749 1/20 0.44
HPN P05981 1/20 0.44
CA1 P00915 1/20 0.43
CA2 P00918 1/20 0.43
MMP1 P03956 1/20 0.43
MMP7 P09237 1/20 0.43
RAB9A P51151 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6571626 1.00 MMP9 (0.65) MMP9MMP2ITGB3ITGA2BTDP1
Hydrochloric Acid SCHEMBL14059215 0.99 MMP9 (0.64) MMP9MMP2ITGB3ITGA2BTDP1
SCHEMBL457772 0.92 MMP9 (0.76) MMP9MMP2ITGB3ITGA2BTDP1
SCHEMBL8001084 0.92 MMP9 (0.76) MMP9MMP2ITGB3ITGA2BTDP1
SCHEMBL10585071 0.92 MMP9 (0.76) MMP9MMP2ITGB3ITGA2BTDP1
SCHEMBL8322406 0.91 MMP9 (0.71) MMP9MMP2ITGB3ITGA2BTDP1
Hydrochloric Acid SCHEMBL9087107 0.91 MMP9 (0.74) MMP9MMP2ITGB3ITGA2BTDP1
SCHEMBL77677 0.90 MMP9 (0.67) MMP9MMP2ITGB3ITGA2BTDP1
SCHEMBL2038720 0.90 MMP9 (0.67) MMP9MMP2ITGB3ITGA2BTDP1
SCHEMBL232590 0.90 MMP9 (0.70) MMP9MMP2ITGB3ITGA2BTDP1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 234 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-10307505-B2 Wound dressings for the controlled release of therapeutic agents KCI USA, INC. (US) 2019-06-04 US claimed
US-20170333592-A1 Wound Dressings For The Controlled Release Of Therapeutic Agents SYSTAGENIX WOUND MANAGEMENT, LIMITED (GB) 2017-11-23 US claimed
US-9687581-B2 Wound dressings for the controlled release of therapeutic agents KCI USA, INC. (US) 2017-06-27 US claimed
CN-105044335-B Immunochromatographic test strip for rapid detection of ancylostomiasis infection and preparation method thereof 中国疾病预防控制中心寄生虫病预防控制所 2017-01-25 CN claimed
CN-105044335-A Immunochromatographic test strip for rapid detection of ancylostomiasis infection and preparation method thereof NAT INST OF PARASITIC DISEASES CHINESE CT FOR DISEASE CONTROL AND PREVENTION 2015-11-11 CN claimed
US-20150098985-A1 WOUND DRESSINGS FOR THE CONTROLLED RELEASE OF THERAPEUTIC KCI USA, INC. 2015-04-09 US claimed
EP-1687039-B1 WOUND DRESSINGS FOR THE CONTROLLED RELEASE OF THERAPEUTIC AGENTS ETHICON INC (US) 2009-01-28 EP claimed
US-20080171691-A1 Inhibition of invasive remodelling LUND LEIF ROGE 2008-07-17 US claimed
EP-0720657-B1 BIOLOGICALLY RELEVANT METHODS FOR THE RAPID DETERMINATION OF STERILITY 3M INNOVATIVE PROPERTIES CO (US) 2007-08-15 EP claimed
US-20070148214-A1 Wound dressing for the controlled release of therapeutic agents KCI USA, INC. 2007-06-28 US claimed
EP-1687039-A1 WOUND DRESSINGS FOR THE CONTROLLED RELEASE OF THERAPEUTIC AGENTS ETHICON, INC. (US) 2006-08-09 EP claimed
US-20050137121-A1 Inhibiting or abolishing the protein cleaving action of plasmin, and inhibiting or abolishing the protein cleaving action of a murine metalloprotease. LUND LEIF R (DK) 2005-06-23 US claimed
WO-2005051441-A1 WOUND DRESSINGS FOR THE CONTROLLED RELEASE OF THERAPEUTIC AGENTS ETHICON, INC. (US) 2005-06-09 WO claimed
EP-0942746-B1 INHIBITION OF INVASIVE REMODELLING FONDEN TIL FREMME AF EKSPERIME (DK) 2005-03-16 EP claimed
US-20020099004-A1 Inhibition of invasive remodelling LUND LEIF ROGE (DK) 2002-07-25 US claimed
US-6180402-B1 REDUCING SIDE EFFECTS OR ENHANCING SELECTIVITY OF THERAPY BY CONTACTING LIVING CELLS WITH PHOTOSENSITIZING AGENT AND AT LEAST ONE CYSTEINE OR SERINE PROTEASE INHIBITOR QLT INC. (CA) 2001-01-30 US claimed
US-6121421-A SIMPLE, EFFICIENT TWO STEP EXTRACTION PROCESS; MIXING CRUDE PREPARATION WITH BUFFER IN WHICH BETA-CASEIN IS INSOLUBLE, PELLETING BETA-CASEIN BY CENTRIFUGING, SUSPENDING PELLET IN BUFFER AND SOLUBILIZER, CENTRIFUGING, SUPERNATANT HAS CASEIN ABBOTT LABORATORIES (US) 2000-09-19 US claimed
WO-1998022098-A2 CPP32 INHIBITORS FOR REGULATING APOPTOSIS QLT PHOTOTHERAPEUTICS, INC. (CA) 1998-05-28 WO claimed
US-4677069-A Clam derived proteinases CORNELL RESEARCH FOUNDATION, INC. (US) 1987-06-30 US claimed
US-12551475-B2 Methods and compositions for treating RNA viral infections MODEL MEDICINES, INC. (US) 2026-02-17 US disclosed
EP-4667008-A2 METHODS AND COMPOSITIONS FOR TREATING RNA VIRAL INFECTIONS Model Medicines, Inc. (US) 2025-12-24 EP disclosed
EP-4000905-B1 PUNCTURE SEALANT SUMITOMO RUBBER IND (JP) 2025-04-09 EP disclosed
US-20250025454-A1 USE OF PIPENDOXIFENE TO TREAT SARS-COV-2 INFECTION MODEL MEDICINES INC (US) 2025-01-23 US disclosed
WO-2024103215-A1 PHARMACEUTICAL COMBINATION FOR TREATING FATTY LIVER DISEASE AND USE THEREOF 泽生生技股份有限公司 2024-05-23 WO disclosed
US-20240082228-A1 SARS-COV-2 THERAPEUTICS MODEL MEDICINES INC (US) 2024-03-14 US disclosed
EP-4281180-A1 SARS-COV-2 THERAPEUTICS Model Medicines, Inc. (US) 2023-11-29 EP disclosed
US-20230346792-A1 COMPOSITIONS AND METHODS FOR TREATING LUNG INFLAMMATION HOTH THERAPEUTICS, INC. 2023-11-02 US disclosed
US-11732113-B2 Puncture sealant SUMITOMO RUBBER INDUSTRIES, LTD. (JP) 2023-08-22 US disclosed
US-20230248712-A1 METHODS AND COMPOSITIONS FOR TREATING RNA VIRAL INFECTIONS MODEL MEDICINES, INC. 2023-08-10 US disclosed
WO-2023102381-A1 USE OF PIPENDOXIFENE TO TREAT SARS-COV-2 INFECTION MODEL MEDICINES, INC. (US) 2023-06-08 WO disclosed
EP-4181928-A1 COMPOSITIONS AND METHODS FOR TREATING LUNG INFLAMMATION Hoth Therapeutics, Inc. (US) 2023-05-24 EP disclosed
EP-4157448-A1 METHODS AND COMPOSITIONS FOR TREATING RNA VIRAL INFECTIONS Model Medicines, Inc. (US) 2023-04-05 EP disclosed
EP-4135660-A1 COMPOSITIONS AND METHODS TO REDUCE THE INFECTIVITY OF A VIRUS Atossa Therapeutics, Inc. (US) 2023-02-22 EP disclosed
WO-2022159763-A1 SARS-COV-2 THERAPEUTICS MODEL MEDICINES, INC. (US) 2022-07-28 WO disclosed
EP-4000905-A1 PUNCTURE SEALANT Sumitomo Rubber Industries, Ltd. (JP) 2022-05-25 EP disclosed
US-20220153965-A1 PUNCTURE SEALANT SUMITOMO RUBBER INDUSTRIES, LTD. (JP) 2022-05-19 US disclosed
WO-2021211808-A1 COMPOSITIONS AND METHODS TO REDUCE THE INFECTIVITY OF A VIRUS ATOSSA THERAPEUTICS, INC. (US) 2021-10-21 WO disclosed
US-20210223258-A9 Method For Protein Kinase Activity Ranking KINOMICA LIMITED (GB) 2021-07-22 US disclosed
EP-3829572-A1 USE OF NEUROKININ-1 ANTAGONISTS TO TREAT CHRONIC PRURITUS Vyne Therapeutics Inc. (US) 2021-06-09 EP disclosed
US-11000535-B2 Anticancer composition and use thereof KAOHSIUNG MEDICAL UNIVERSITY (TW) 2021-05-11 US disclosed
US-10870885-B2 Dendritic cell response gene expression, compositions of matters and methods of use thereof THE BROAD INSTITUTE, INC. (US) 2020-12-22 US disclosed
EP-3627153-B1 A METHOD OF ASSESSING PROTEIN MODIFICATION STATUS AND IDENTIFYING BIOMARKERS LINKED TO CELL SIGNALING PATHWAYS UNIV LONDON QUEEN MARY (GB) 2020-10-07 EP disclosed
EP-3377905-B1 METHOD FOR PROTEIN KINASE ACTIVITY RANKING UNIV LONDON QUEEN MARY (GB) 2020-09-02 EP disclosed
US-20200249239-A1 Method For Protein Kinase Activity Ranking UNIV LONDON QUEEN MARY (GB) 2020-08-06 US disclosed
US-20200221753-A1 TEXTURED INGESTIBLE PRODUCTS EETBE INC (US) 2020-07-16 US disclosed
EP-2224000-B1 ANTIBODY AND USE THEREOF TAO HEALTH LIFE PHARMA CO LTD (JP) 2020-05-13 EP disclosed
EP-3627153-A1 A METHOD OF ASSESSING PROTEIN MODIFICATION STATUS AND IDENTIFYING BIOMARKERS LINKED TO CELL SIGNALING PATHWAYS Queen Mary University of London (GB) 2020-03-25 EP disclosed
WO-2020023898-A1 USE OF NEUROKININ-1 ANTAGONISTS TO TREAT CHRONIC PRURITUS MENLO THERAPEUTICS INC. (US) 2020-01-30 WO disclosed
EP-3304075-B1 A METHOD OF ASSESSING PROTEIN MODIFICATION STATUS AND IDENTIFYING BIOMARKERS LINKED TO CELL SIGNALING PATHWAYS UNIV LONDON QUEEN MARY (GB) 2019-08-21 EP disclosed
US-20190216779-A1 USE OF NEUROKININ-1 ANTAGONISTS TO TREAT A VARIETY OF PRURITIC CONDITIONS MENLO THERAPEUTICS INC. (US) 2019-07-18 US disclosed
US-10307505-B2 Wound dressings for the controlled release of therapeutic agents KCI USA, INC. (US) 2019-06-04 US disclosed
EP-3478283-A1 USE OF NEUROKININ-1 ANTAGONISTS TO TREAT A VARIETY OF PRURITIC CONDITIONS Menlo Therapeutics Inc. (US) 2019-05-08 EP disclosed
EP-3377905-A1 METHOD FOR PROTEIN KINASE ACTIVITY RANKING Queen Mary University of London (GB) 2018-09-26 EP disclosed
US-20180235931-A1 USE OF NEUROKININ-1 ANTAGONISTS AS ANTITUSSIVES MENLO THERAPEUTICS INC. 2018-08-23 US disclosed
US-20180214469-A1 ANTICANCER COMPOSITION AND USE THEREOF KAOHSIUNG MEDICAL UNIVERSITY (TW) 2018-08-02 US disclosed
US-20180217129-A1 A Method Of Assessing Protein Modification Status And Identifying Biomarkers Linked To Cell Signaling Pathways QUEEN MARY UNIVERSITY OF LONDON (GB) 2018-08-02 US disclosed
WO-2018136554-A1 USE OF NEUROKININ-1 ANTAGONISTS AS ANTITUSSIVES MENLO THERAPEUTICS INC. (US) 2018-07-26 WO disclosed
US-9993425-B2 Compositions for intranasal delivery of human insulin and uses thereof MARINA BIOTECH, INC. (US) 2018-06-12 US disclosed
EP-3304075-A1 A METHOD OF ASSESSING PROTEIN MODIFICATION STATUS AND IDENTIFYING BIOMARKERS LINKED TO CELL SIGNALING PATHWAYS Queen Mary University of London (GB) 2018-04-11 EP disclosed
US-20180000930-A1 Methods and Compositions for Preserving the Viability of Photoreceptor Cells MASSACHUSETTS EYE & EAR INFIRMARY (US) 2018-01-04 US disclosed
WO-2018005695-A1 USE OF NEUROKININ-1 ANTAGONISTS TO TREAT A VARIETY OF PRURITIC CONDITIONS MENLO THERAPEUTICS INC. (US) 2018-01-04 WO disclosed
US-9840731-B2 Preservation of biological materials in non-aqueous fluid media GENTEGRA, LLC (US) 2017-12-12 US disclosed
US-20170333592-A1 Wound Dressings For The Controlled Release Of Therapeutic Agents SYSTAGENIX WOUND MANAGEMENT, LIMITED (GB) 2017-11-23 US disclosed
US-9782464-B2 Methods and compositions for inhibiting diseases of the central nervous system BOARD OF REGENTS OF THE UNIVERSITY OF NEBRASKA (US) 2017-10-10 US disclosed
US-20170196253-A1 TEXTURED INGESTIBLE PRODUCTS EETBE, INC. 2017-07-13 US disclosed
US-20170196806-A1 METHODS AND COMPOSITIONS FOR PRESERVING THE VIABILITY OF PHOTORECEPTOR CELLS MASSACHUSETTS EYE & EAR INFIRMARY (US) 2017-07-13 US disclosed
US-9687581-B2 Wound dressings for the controlled release of therapeutic agents KCI USA, INC. (US) 2017-06-27 US disclosed
CN-106714544-A Textured ingestible products 埃特比公司 2017-05-24 CN disclosed
CN-105044335-B Immunochromatographic test strip for rapid detection of ancylostomiasis infection and preparation method thereof 中国疾病预防控制中心寄生虫病预防控制所 2017-01-25 CN disclosed
US-9549895-B2 Methods and compositions for preserving the viability of photoreceptor cells MASSACHUSETTS EYE AND EAR INFIRMARY (US) 2017-01-24 US disclosed
WO-2016193745-A1 A METHOD OF ASSESSING PROTEIN MODIFICATION STATUS AND IDENTIFYING BIOMARKERS LINKED TO CELL SIGNALING PATHWAYS QUEEN MARY UNIVERSITY OF LONDON (GB) 2016-12-08 WO disclosed
US-20160184417-A1 Methods and Compositions for Inhibiting Diseases of the Central Nervous System BOARD OF REGENTS OF THE UNIVERSITY OF NEBRASKA 2016-06-30 US disclosed
US-20160144024-A1 Methods and Compositions for Preserving the Viability of Photoreceptor Cells MASSACHUSETTS EYE AND EAR INFIRMARY 2016-05-26 US disclosed
US-9259465-B2 Methods and compositions for inhibiting diseases of the central nervous system BOARD OF REGENTS OF THE UNIVERSITY OF NEBRASKA (US) 2016-02-16 US disclosed
EP-2971116-A1 DENDRITIC CELL RESPONSE GENE EXPRESSION, COMPOSITIONS OF MATTERS AND METHODS OF USE THEREOF The Broad Institute, Inc. (US) 2016-01-20 EP disclosed
US-20150368719-A1 DENDRITIC CELL RESPONSE GENE EXPRESSION, COMPOSITIONS OF MATTERS AND METHODS OF USE THEREOF THE BROAD INSTITUTE, INC. 2015-12-24 US disclosed
US-9212387-B2 Method for detection of genes targeted by microRNA NATIONAL UNIVERSITY CORPORATION OKAYAMA UNIVERSITY (JP) 2015-12-15 US disclosed
CN-105044335-A Immunochromatographic test strip for rapid detection of ancylostomiasis infection and preparation method thereof NAT INST OF PARASITIC DISEASES CHINESE CT FOR DISEASE CONTROL AND PREVENTION 2015-11-11 CN disclosed
US-20150297619-A1 METHODS AND COMPOSITIONS FOR PRESERVING THE MUCOSAL BARRIER THE REGENTS OF THE UNIVERSITY OF CALIFORNIA 2015-10-22 US disclosed
US-20150267245-A1 PRESERVATION OF BIOLOGICAL MATERIALS IN NON-AQUEOUS FLUID MEDIA GENTEGRA, LLC (US) 2015-09-24 US disclosed
US-20150098985-A1 WOUND DRESSINGS FOR THE CONTROLLED RELEASE OF THERAPEUTIC KCI USA, INC. 2015-04-09 US disclosed
EP-2846788-A1 USE OF COMPOUNDS FOR THE TREATMENT OF PAIN Akron Molecules AG (AT) 2015-03-18 EP disclosed
WO-2014197090-A2 PRESERVATION OF BIOLOGICAL MATERIALS IN NON-AQUEOUS FLUID MEDIA GENTEGRA, LLC (US) 2014-12-11 WO disclosed
US-20140349969-A1 COMPOUNDS AND METHODS FOR TREATING PAIN AKRON MOLECULES AG (AT) 2014-11-27 US disclosed
EP-2584046-B1 METHOD FOR DETECTION OF GENES TARGETED BY MICRORNA UNIV OKAYAMA NAT UNIV CORP (JP) 2014-11-19 EP disclosed
US-8858987-B2 Wound dressing for the controlled release of therapeutic agents SYSTAGENIX WOUND MANAGEMENT (US), INC. (US) 2014-10-14 US disclosed
EP-2780029-A1 ORAL LEPTIN FORMULATIONS AND USES THEREOF Université de Montréal (CA) 2014-09-24 EP disclosed
WO-2014145631-A1 DENDRITIC CELL RESPONSE GENE EXPRESSION, COMPOSITIONS OF MATTERS AND METHODS OF USE THEREOF THE BROAD INSTITUTE, INC. (US) 2014-09-18 WO disclosed
WO-2014055936-A1 PRESERVATION OF BIOLOGICAL MATERIALS IN NON-AQUEOUS FLUID MEDIA INTEGENX INC. (US) 2014-04-10 WO disclosed
US-20140004148-A1 Methods and Compositions for Inhibiting Diseases of the Central Nervous System NATIONAL INSTITUTES OF HEALTH (NIH), U.S. DEPT. OF HEALTH AND HUMAN SERVICES (DHHS), U.S. GOVERNMENT 2014-01-02 US disclosed
EP-2674161-A1 FMO3 inhibitors for treating pain Akron Molecules GmbH (AT) 2013-12-18 EP disclosed
CN-103415286-A Compounds and methods for treating pain AKRON MOLECULES GMBH 2013-11-27 CN disclosed
WO-2013167743-A1 USE OF COMPOUNDS FOR THE TREATMENT OF PAIN AKRON MOLECULES GMBH (AT) 2013-11-14 WO disclosed
US-20130252924-A1 Compounds and Methods for Treating Pain AKRON MOLECULES GMBH (AT) 2013-09-26 US disclosed
EP-2637649-A2 COMPOUNDS AND METHODS FOR TREATING PAIN Akron Molecules GmbH (AT) 2013-09-18 EP disclosed
US-20130224110-A1 USE OF ADENOSINE RECEPTOR SIGNALING TO MODULATE PERMEABILITY OF BLOOD-BRAIN BARRIER CORNELL UNIVERSITY (US) 2013-08-29 US disclosed
US-20130217050-A1 METHOD FOR DIAGNOSING ALZHEIMER'S DISEASE USING-SOLUBLE GPVI MOCHIDA PHARMACEUTICAL CO., LTD. (JP) 2013-08-22 US disclosed
EP-2616538-A1 USE OF ADENOSINE RECEPTOR SIGNALING TO MODULATE PERMEABILITY OF BLOOD-BRAIN BARRIER Cornell University (US) 2013-07-24 EP disclosed
US-8491890-B2 Methods and compositions for inhibiting diseases of the central nervous system BOARD OF REGENTS OF THE UNIVERSITY OF NEBRASKA (US) 2013-07-23 US disclosed
EP-2615458-A1 METHOD FOR DIAGNOSING ALZHEIMER'S DISEASE USING BLOOD-SOLUBLE GPVI Mochida Pharmaceutical Co., Ltd. (JP) 2013-07-17 EP disclosed
WO-2013071396-A1 ORAL LEPTIN FORMULATIONS AND USES THEREOF Université de Montréal (CA) 2013-05-23 WO disclosed
US-8445649-B2 Antibody and use thereof TAO HEALTH LIFE PHARMA CO., LTD. (JP) 2013-05-21 US disclosed
EP-2584046-A1 KIT FOR DETECTION OF GENES TARGETED BY MICRORNA, AND METHOD FOR DETECTION OF GENES TARGETED BY MICRORNA National University Corporation Okayama University (JP) 2013-04-24 EP disclosed
US-20130089866-A1 Kit For Detection of Genes Targeted by MicroRNA, and Method For Detection of Genes Targeted by MicroRNA NATIONAL UNIVERSITY CORPORATION OKAYAMA UNIVERSITY (JP) 2013-04-11 US disclosed
WO-2012062925-A2 COMPOUNDS AND METHODS FOR TREATING PAIN AKRON MOLECULES GMBH (AT) 2012-05-18 WO disclosed
US-8168188-B1 Antibody and utilization of the same KYOTO UNIVERSITY (JP) 2012-05-01 US disclosed
US-20120094903-A1 COMPOSITIONS FOR INTRANASAL DELIVERY OF HUMAN INSULIN AND USES THEREOF MARINA BIOTECH INC. (US) 2012-04-19 US disclosed
WO-2012037457-A1 USE OF ADENOSINE RECEPTOR SIGNALING TO MODULATE PERMEABILITY OF BLOOD-BRAIN BARRIER CORNELL UNIVERSITY (US) 2012-03-22 WO disclosed
CN-101340893-B Intranasal administration of rapid acting insulin NASTECH PHARM CO 2012-03-21 CN disclosed
US-20110159004-A1 Methods and Compositions for Preserving the Viability of Photoreceptor Cells MASSACHUSETTS EYE AND EAR INFIRMARY 2011-06-30 US disclosed
US-7863245-B2 Compositions for enhanced epithelial permeation of neuropeptide Y for treating obesity NASTECH PHARMACEUTICAL COMPANY, INC. (US) 2011-01-04 US disclosed
US-20100297662-A1 ANTIBODY AND USE THEREOF FOUNDATION FOR BIOMEDICAL RESEARCH AND INNOVATION AT KOBE (JP) 2010-11-25 US disclosed
US-7811832-B2 Methods for preserving the viability of photoreceptor cells by anti-FAS-ligand/anti-FAS-receptor antibodies MASSACHUSETTS EYE AND EAR INFIRMARY (US) 2010-10-12 US disclosed
EP-1696960-B1 INTRANASAL ADMINISTRATION OF GLUCOSE-REGULATING PEPTIDES AMYLIN PHARMACEUTICALS INC (US) 2010-09-08 EP disclosed
EP-2224000-A1 ANTIBODY AND USE THEREOF Kyoto University (JP) 2010-09-01 EP disclosed
US-20100210506-A1 INTRANASAL ADMINISTRATION OF RAPID ACTING INSULIN MDRNA, INC. (US) 2010-08-19 US disclosed
EP-1951198-B1 INTRANASAL ADMINISTRATION OF RAPID ACTING INSULIN MDRNA INC (US) 2010-06-16 EP disclosed
US-20100074882-A1 METHODS AND COMPOSITIONS FOR PRESERVING THE VIABILITY OF PHOTORECEPTOR CELLS NATIONAL INSTITUTES OF HEALTH - DIRECTOR DEITR 2010-03-25 US disclosed
US-20100028320-A1 Methods and Compositions for Inhibiting Diseases of the Central Nervous System BOARD OF REGENTS OF THE UNIVERSITY OF NEBRASKA 2010-02-04 US disclosed
US-20090325860-A1 COMPOSITIONS FOR INTRANASAL DELIVERY OF HUMAN INSULIN AND USES THEREOF NASTECH PHARMACEUTICAL COMPANY INC. (US) 2009-12-31 US disclosed
CN-100569281-C Preparation and use of composition for treating and preventing necrosis ILANA NATHAN (IL) 2009-12-16 CN disclosed
US-7592330-B2 Methods and compositions for preserving the viability of photoreceptor cells MASSACHUSETTS EYE AND EAR INFIRMARY (US) 2009-09-22 US disclosed
US-20090118158-A1 COMPOSITIONS FOR ENHANCED EPITHELIAL PERMEATION OF PEPTIDE YY FOR TREATING OBESITY NASTECH PHARMACEUTICAL COMPANY INC. (US) 2009-05-07 US disclosed
EP-2046284-A1 COMPOSITIONS FOR INTRANASAL DELIVERY OF HUMAN INSULIN AND USES THEREOF Nastech Pharmaceutical Company Inc. (US) 2009-04-15 EP disclosed
US-20090054326-A1 FORMULATIONS FOR ENHANCED MUCOSAL DELIVERY OF PYY NASTECH PHARMACEUTICAL COMPANY INC. (US) 2009-02-26 US disclosed
EP-1687039-B1 WOUND DRESSINGS FOR THE CONTROLLED RELEASE OF THERAPEUTIC AGENTS ETHICON INC (US) 2009-01-28 EP disclosed
CN-101340893-A Intranasal administration of rapid acting insulin NASTECH PHARM CO (US) 2009-01-07 CN disclosed
US-20080318837-A1 Pharmaceutical Formation For Increased Epithelial Permeability of Glucose-Regulating Peptide NASTECH PHARMACEUTICAL COMPANY INC. (US) 2008-12-25 US disclosed
US-20080318861-A1 Mucosal Delivery of Stabilized Formulations of Exendin NASTECH PHARMACEUTICAL COMPANY INC. (US) 2008-12-25 US disclosed
US-20080234200-A1 Saline formulation of a glucose-regulating peptide (amylin, synthtic hormone pramlintide, glucon like peptide-1, extendins), water, sodium chloride and a buffering agent; identical ph and osmolarity for both transmucosal glucose regulating peptide and saline water; antidiabetic, antiobesity agent NASTECH PHARMACEUTICAL COMPANY INC. (US) 2008-09-25 US disclosed
EP-1965828-A2 PHARMACEUTICAL FORMULATION FOR INCREASED EPITHELIAL PERMEABILITY OF GLUCOSE-REGULATING PEPTIDE Nastech Pharmaceutical Company Inc. (US) 2008-09-10 EP disclosed
CN-101262888-A Formulations for enhanced mucosal delivery of PYY NASTECH PHARM CO (US) 2008-09-10 CN disclosed
EP-1959987-A2 MUCOSAL DELIVERY OF STABILIZED FORMULATIONS OF EXENDIN Nastech Pharmaceutical Company Inc. (US) 2008-08-27 EP disclosed
EP-1951198-A2 INTRANASAL ADMINISTRATION OF RAPID ACTING INSULIN Nastech Pharmaceutical Company Inc. (US) 2008-08-06 EP disclosed
US-20080171691-A1 Inhibition of invasive remodelling LUND LEIF ROGE 2008-07-17 US disclosed
US-20080113011-A1 Compositions and methods for enhanced mucosal delivery of interferon beta NASTECH PHARMACEUTICAL COMPANY INC. (US) 2008-05-15 US disclosed
EP-1664719-A4 METHODS FOR SUBSTANTIALLY SIMULTANEOUS EVALUATION OF A SAMPLE CONTAINING A CELLULAR TARGET AND A SOLUBLE ANALYTE BECKMAN COULTER INC (US) 2008-04-09 EP disclosed
EP-1907008-A2 FORMULATIONS FOR ENHANCED MUCOSAL DELIVERY OF PYY Nastech Pharmaceutical Company Inc. (US) 2008-04-09 EP disclosed
EP-1539220-A4 COMPOSITIONS AND METHODS FOR ENHANCED MUCOSAL DELIVERY OF INTERFERON BETA NASTECH PHARM CO (US) 2008-04-02 EP disclosed
WO-2008016729-A1 COMPOSITIONS FOR INTRANASAL DELIVERY OF HUMAN INSULIN AND USES THEREOF NASTECH PHARMACEUTICAL COMPANY INC. (US) 2008-02-07 WO disclosed
US-20080004218-A1 METHODS FOR ENHANCED EPITHELIAL PERMEATION OF Y2 RECEPTOR-BINDING PEPTIDES FOR TREATING AND PREVENTING OBESITY NASTECH PHARMACEUTICAL COMPANY INC. 2008-01-03 US disclosed
WO-2007146448-A1 PHARMACEUTICAL FORMULATIONS OF GLP-1 DERIVATIVES NASTECH PHARMACEUTICAL COMPANY INC. (US) 2007-12-21 WO disclosed
US-20070287756-A1 Methods and Compositions for Preserving the Viability of Photoreceptor Cells MASSACHUSETTS EYE AND EAR INFIRMARY 2007-12-13 US disclosed
US-20070275893-A1 COMPOSITIONS FOR ENHANCED EPITHELIAL PERMEATION OF PEPTIDE YY FOR TREATING OBESITY NASTECH PHARMACEUTICAL COMPANY INC. 2007-11-29 US disclosed
CN-101080421-A Antibody and use thereof MITSUBISHI CHEM CORP (JP) 2007-11-28 CN disclosed
US-20070232537-A1 INTRANASAL PYY FORMULATIONS WITH IMPROVED TRANSMUCOSAL PHARMACOKINETICS NASTECH PHARMACEUTICAL COMPANY INC. (US) 2007-10-04 US disclosed
US-20070213270-A1 PEPTIDE YY FORMULATIONS HAVING INCREASED STABILITY AND RESISTANCE TO MICROBIAL AGENTS NASTECH PHARMACEUTICAL COMPANY INC. 2007-09-13 US disclosed
US-20070197437-A1 COMPOSITIONS FOR ENHANCED EPITHELIAL PERMEATION OF Y2 RECEPTOR-BINDING PEPTIDES NASTECH PHARMACEUTICAL COMPANY INC. 2007-08-23 US disclosed
EP-0720657-B1 BIOLOGICALLY RELEVANT METHODS FOR THE RAPID DETERMINATION OF STERILITY 3M INNOVATIVE PROPERTIES CO (US) 2007-08-15 EP disclosed
US-20070185035-A1 ENHANCED MUCOSAL ADMINISTRATION OF NEUROPROTECTIVE PEPTIDES NASTECH PHARMACEUTICAL COMPANY INC. (US) 2007-08-09 US disclosed
US-20070161563-A1 A DEVICE FOR ENHANCED EPITHELIAL PERMEATION OF Y2 RECEPTOR-BINDING PEPTIDES NASTECH PHARMACEUTICAL COMPANY INC. 2007-07-12 US disclosed
US-20070148214-A1 Wound dressing for the controlled release of therapeutic agents KCI USA, INC. 2007-06-28 US disclosed
WO-2007067964-A2 MUCOSAL DELIVERY OF STABILIZED FORMULATIONS OF EXENDIN NASTECH PHARMACEUTICAL COMPANY INC. (US) 2007-06-14 WO disclosed
US-7229966-B2 Compositions and methods for enhanced mucosal delivery of Y2 receptor-binding peptides and methods for treating and preventing obesity NASTECH PHARMACEUTICAL COMPANY INC. (US) 2007-06-12 US disclosed
WO-2007065156-A2 PHARMACEUTICAL FORMULATION FOR INCREASED EPITHELIAL PERMEABILITY OF GLUCOSE-REGULATING PEPTIDE NASTECH PHARMACEUTICAL COMPANY INC. (US) 2007-06-07 WO disclosed
US-20070129299-A1 COMPOSITIONS AND METHODS FOR ENHANCED MUCOSAL DELIVERY OF PYY PEPTIDE NASTECH PHARMACEUTICAL COMPANY INC. 2007-06-07 US disclosed
WO-2007061434-A2 A PHARMACEUTICAL FORMULATION OF GLP-1 AND ITS USE FOR TREATING A METABOLIC SYNDROME NASTECH PHARMACEUTICAL COMPANY INC. (US) 2007-05-31 WO disclosed
EP-1787998-A1 ANTIBODY AND UTILIZATION OF THE SAME Mitsubishi Chemical Corporation (JP) 2007-05-23 EP disclosed
WO-2007047948-A2 INTRANASAL ADMINISTRATION OF RAPID ACTING INSULIN NASTECH PHARMACEUTICAL COMPANY INC. (US) 2007-04-26 WO disclosed
US-20070077283-A1 METHOD OF ENHANCING TRANSMUCOSAL DELIVERY OF THERAPEUTIC COMPOUNDS NASTECH PHARMACEUTICAL COMPANY INC. 2007-04-05 US disclosed
US-7186691-B2 Compositions and methods for enhanced mucosal delivery of Y2 receptor-binding peptides and methods for treating and preventing obesity NASTECH PHARMACEUTICAL COMPANY INC. (US) 2007-03-06 US disclosed
US-7186692-B2 Compositions and methods for enhanced mucosal delivery and non-infused administration of Y2 receptor-binding peptides and methods for treating and preventing obesity NASTECH PHARMACEUTICAL COMPANY INC. (US) 2007-03-06 US disclosed
WO-2007019427-A2 METHODS AND COMPOSITIONS FOR PRESERVING THE VIABILITY OF PHOTORECEPTOR CELLS MASSACHUSETTS EYE & EAR INFIRMARY (US) 2007-02-15 WO disclosed
US-20070032427-A1 Methods and compositions for preserving the viability of photoreceptor cells MASSACHUSETTS EYE AND EAR INFIRMARY 2007-02-08 US disclosed
US-7166575-B2 Compositions and methods for enhanced mucosal delivery of peptide YY and methods for treating and preventing obesity NASTECH PHARMACEUTICAL COMPANY INC. (US) 2007-01-23 US disclosed
WO-2007008778-A2 FORMULATIONS FOR ENHANCED MUCOSAL DELIVERY OF PYY NASTECH PHARMACEUTICAL COMPANY INC. (US) 2007-01-18 WO disclosed
US-7157426-B2 such as peptide YY, Neuropeptide Y, or Pancreatic polypeptide with solubilizing agent (cyclodextran), chelating agent (ethylenediamine tetraacetic acid), and polyol such as sucrose NASTECH PHARMACEUTICAL COMPANY INC. (US) 2007-01-02 US disclosed
EP-1715885-A2 COMPOSITIONS AND METHODS FOR ENHANCED MUCOSAL DELIVERY OF Y2 RECEPTOR-BINDING PEPTIDES AND METHODS FOR TREATING AND PREVENTING OBESITY Nastech Pharmaceutical Company Inc. (US) 2006-11-02 EP disclosed
WO-2006007412-A9 PEPTIDE YY FORMULATIONS HAVING INCREASED STABILITY AND RESISTANCE TO MICROBIAL AGENTS NASTECH PHARM CO (US) 2006-09-21 WO disclosed
US-20060210614-A1 Mucosal delivery-enhancing agent selected from a solubilization agent; a charge-modifying agent; a pH control agent; a degradative enzyme inhibitor; a mucolytic/mucus clearing agent; increased bioavailability of exendins peptide when administered intranasally to a mammal; antidiabetic/antiobesity agent NASTECH PHARMACEUTICAL COMPANY INC. 2006-09-21 US disclosed
EP-1696960-A1 INTRANASAL ADMINISTRATION OF GLUCOSE-REGULATING PEPTIDES Nastech Pharmaceutical Company Inc. (US) 2006-09-06 EP disclosed
EP-1687039-A1 WOUND DRESSINGS FOR THE CONTROLLED RELEASE OF THERAPEUTIC AGENTS ETHICON, INC. (US) 2006-08-09 EP disclosed
EP-1664719-A2 METHODS FOR SUBSTANTIALLY SIMULTANEOUS EVALUATION OF A SAMPLE CONTAINING A CELLULAR TARGET AND A SOLUBLE ANALYTE Beckman Coulter, Inc. (US) 2006-06-07 EP disclosed
US-20060074025-A1 Therapeutic formulations for transmucosal administration that increase glucagon-like peptide-1 bioavailability NASTECH PHARMACEUTICAL COMPANY INC. 2006-04-06 US disclosed
US-20060069021-A1 Compositions and methods for intranasal administration of inactive analogs of PTH or inactivated preparations of PTH or PTH analogs NASTECH PHARMACEUTICAL COMPANY INC. 2006-03-30 US disclosed
US-20060024744-A1 Methods for substantially simultaneous evaluation of a sample containing a cellular target and a soluble analyte BECKMAN COULTER, INC. 2006-02-02 US disclosed
WO-2006007412-A2 PEPTIDE YY FORMULATIONS HAVING INCREASED STABILITY AND RESISTANCE TO MICROBIAL AGENTS NASTECH PHARMACEUTICAL COMPANY INC. (US) 2006-01-19 WO disclosed
WO-2005105133-A2 METHODS AND COMPOSITIONS FOR PRESERVING THE VIABILITY OF PHOTORECEPTOR CELLS MASSACHUSETTS EYE AND EAR INFIRMARY (US) 2005-11-10 WO disclosed
EP-1581245-A2 COMPOSITIONS AND METHODS FOR ENHANCED MUCOSAL DELIVERY OF Y2 RECEPTOR-BINDING PEPTIDES AND METHODS FOR TREATING AND PREVENTING OBESITY Nastech Pharmaceutical Company Inc. (US) 2005-10-05 EP disclosed
WO-2005080433-A2 COMPOSITIONS AND METHODS FOR ENHANCED MUCOSAL DELIVERY OF Y2 RECEPTOR-BINDING PEPTIDES AND METHODS FOR TREATING AND PREVENTING OBESITY NASTECH PHARMACEUTICAL COMPANY INC. (US) 2005-09-01 WO disclosed
WO-2005075015-A1 TREATMENT DEVICE FOR WOUND THERAPY ETHICON, INC. (US) 2005-08-18 WO disclosed
CN-1655809-A Compositions and methods for treating and preventing necrosis ILANA NATHAN (IL) 2005-08-17 CN disclosed
WO-2005065714-A1 INTRANASAL ADMINISTRATION OF GLUCOSE-REGULATING PEPTIDES NASTECH PHARMACEUTICAL COMPANY INC. (US) 2005-07-21 WO disclosed
US-20050143303-A1 Intranasal administration of glucose-regulating peptides NASTECH PHARMACEUTICAL COMPANY INC. 2005-06-30 US disclosed
US-20050137121-A1 Inhibiting or abolishing the protein cleaving action of plasmin, and inhibiting or abolishing the protein cleaving action of a murine metalloprotease. LUND LEIF R (DK) 2005-06-23 US disclosed
US-20050129684-A1 Methods and compositions for preserving the viability of photoreceptor cells MASSACHUSETTS EYE AND EAR INFIRMARY 2005-06-16 US disclosed
EP-1539220-A2 COMPOSITIONS AND METHOD FOR ENHANCED MUCOSAL DELIVERY OF INTERFERON BETA Nastech Pharmaceutical Company Inc. (US) 2005-06-15 EP disclosed
EP-1539208-A2 COMPOSITIONS AND METHODS FOR MODULATING PHYSIOLOGY OF EPITHELIAL JUNCTIONAL ADHESION MOLECULES FOR ENHANCED MUCOSAL DELIVERY OF THERAPEUTIC COMPOUNDS Nastech Pharmaceutical Company Inc. (US) 2005-06-15 EP disclosed
WO-2005051441-A1 WOUND DRESSINGS FOR THE CONTROLLED RELEASE OF THERAPEUTIC AGENTS ETHICON, INC. (US) 2005-06-09 WO disclosed
WO-2005036123-A2 METHODS FOR SUBSTANTIALLY SIMULTANEOUS EVALUATION OF A SAMPLE CONTAINING A CELLULAR TARGET AND A SOLUBLE ANALYTE BECKMAN COULTER, INC. (US) 2005-04-21 WO disclosed
US-20050069958-A1 Method for simultaneous evaluation of a sample containing a cellular target and a soluble analyte BECKMAN COULTER, INC. 2005-03-31 US disclosed
EP-0942746-B1 INHIBITION OF INVASIVE REMODELLING FONDEN TIL FREMME AF EKSPERIME (DK) 2005-03-16 EP disclosed
US-20050002927-A1 Compositions and methods for enhanced mucosal delivery and non-infused administration of Y2 receptor-binding peptides and methods for treating and preventing obesity NASTECH PHARMACEUTICAL COMPANY INC. (US) 2005-01-06 US disclosed
US-20040214772-A1 Compositions and methods for enhanced mucosal delivery of Y2 receptor-binding peptides and methods for treating and preventing obesity NASTECH PHARMACEUTICAL COMPANY INC. 2004-10-28 US disclosed
US-20040209807-A1 Compositions and methods for enhanced mucosal delivery of Y2 receptor-binding peptides and methods for treating and preventing obesity NASTECH PHARMACEUTICAL COMPANY INC. 2004-10-21 US disclosed
EP-1450764-A2 DOPAMINE AGONIST FORMULATIONS FOR ENHANCED CENTRAL NERVOUS SYSTEM DELIVERY NASTECH PHARMACEUTICAL COMPANY, INC. (US) 2004-09-01 EP disclosed
US-20040157777-A1 Compositions and methods for enhanced mucosal delivery of Y2 receptor-binding peptides and methods for treating and preventing obesity NASTECH PHARMACEUTICAL COMPANY INC. 2004-08-12 US disclosed
EP-0720657-A4 BIOLOGICALLY RELEVANT METHODS FOR THE RAPID DETERMINATION OF STERILITY 3M INNOVATIVE PROPERTIES CO (US) 2004-08-04 EP disclosed
WO-2004056314-A2 COMPOSITIONS AND METHODS FOR ENHANCED MUCOSAL DELIVERY OF Y2 RECEPTOR-BINDING PEPTIDES AND METHODS FOR TREATING AND PREVENTING OBESITY NASTECH PHARMACEUTICAL COMPANY INC. (US) 2004-07-08 WO disclosed
US-20040115135-A1 Compositions and methods for enhanced mucosal delivery of peptide YY and methods for treating and preventing obesity MARINA BIOTECH, INC. 2004-06-17 US disclosed
US-20040077540-A1 Compositions and methods for modulating physiology of epithelial junctional adhesion molecules for enhanced mucosal delivery of therapeutic compounds NASTECH PHARMACEUTICAL COMPANY INC. 2004-04-22 US disclosed
US-20040037809-A1 Compositions and methods for enhanced mucosal delivery of interferon beta NASTECH PHARMACEUTICAL COMPANY INC. 2004-02-26 US disclosed
US-20040028613-A1 Dopamine agonist formulations for enhanced central nervous system delivery NASTECH PHARMACEUTICAL COMPANY INC 2004-02-12 US disclosed
WO-2004002404-A2 COMPOSITIONS AND METHOD FOR ENHANCED MUCOSAL DELIVERY OF INTERFERON BETA NASTECH PHARMACEUTICAL COMPANY INC. (US) 2004-01-08 WO disclosed
WO-2004003145-A2 COMPOSITIONS AND METHODS FOR MODULATING PHYSIOLOGY OF EPITHELIAL JUNCTIONAL ADHESION MOLECULES FOR ENHANCED MUCOSAL DELIVERY OF THERAPEUTIC COMPOUNDS NASTECH PHARMACEUTICAL COMPANY INC. (US) 2004-01-08 WO disclosed
WO-2003000018-A2 DOPAMINE AGONIST FORMULATIONS FOR ENHANCED CENTRAL NERVOUS SYSTEM DELIVERY NASTECH PHARMACEUTICAL COMPANY, INC. (US) 2003-01-03 WO disclosed
US-20020192754-A1 Method for producing active serine proteases and inactive variants MAX-PLANCK-GESELLSCHAFT E.V. (DE) 2002-12-19 US disclosed
EP-0850244-B1 TOXOPLASMA GONDII GLYCOCONJUGATES ORGANON TEKNIKA BV (NL) 2002-07-31 EP disclosed
US-20020099004-A1 Inhibition of invasive remodelling LUND LEIF ROGE (DK) 2002-07-25 US disclosed
CN-1352682-A Cysteine protease and inhibitors for the prevention and treatment of neurocysticercosis UNIV GEORGIA RESAERCH FOUNDATI (US) 2002-06-05 CN disclosed
US-20020058288-A1 Compound for use in the detection and prevention of parasitic infection of humans AKZO NOBEL N.V. (NL) 2002-05-16 US disclosed
US-6180402-B1 REDUCING SIDE EFFECTS OR ENHANCING SELECTIVITY OF THERAPY BY CONTACTING LIVING CELLS WITH PHOTOSENSITIZING AGENT AND AT LEAST ONE CYSTEINE OR SERINE PROTEASE INHIBITOR QLT INC. (CA) 2001-01-30 US disclosed
US-6121421-A SIMPLE, EFFICIENT TWO STEP EXTRACTION PROCESS; MIXING CRUDE PREPARATION WITH BUFFER IN WHICH BETA-CASEIN IS INSOLUBLE, PELLETING BETA-CASEIN BY CENTRIFUGING, SUSPENDING PELLET IN BUFFER AND SOLUBILIZER, CENTRIFUGING, SUPERNATANT HAS CASEIN ABBOTT LABORATORIES (US) 2000-09-19 US disclosed
WO-2000011890-A2 METHODS FOR ISOLATING RECOMBINANT β-CASEIN ABBOTT LABORATORIES (US) 2000-03-02 WO disclosed
US-5976859-A COMPOSITIONS FOR CLEANING AND WASHING PURPOSES. WISCONSIN ALUMNI RESEARCH FOUNDATION (US) 1999-11-02 US disclosed
US-5863742-A LYSING CELLS IN SAMPLE WITH NONIONIC DETERGENT TO RELEASE MX PROTEIN, INACTIVATING PROTEASE BY HEATING WITH DENATURING AGENT, REACTING SOLUTION WITH MONOCLONAL ANTIBODY CLONE, DETECTING BINDING OF ANTIBODY TO PROTEIN CHIRON DIAGNOSTICS CORPORATION (US) 1999-01-26 US disclosed
US-5849988-A Rat comprising straight filaments in its brain TRUSTEES OF THE UNIVERSITY OF PENNSYLVANIA (US) 1998-12-15 US disclosed
EP-0749493-B1 INHIBITION OF PROTEASE ACTIVITY OF HUMAN WHOLE BLOOD CELL LYSATES CIBA CORNING DIAGNOSTICS CORP (US) 1998-09-23 EP disclosed
WO-1998022098-A2 CPP32 INHIBITORS FOR REGULATING APOPTOSIS QLT PHOTOTHERAPEUTICS, INC. (CA) 1998-05-28 WO disclosed
WO-1998021319-A1 DETERGENT-STABLE MICROBIAL PROTEASE WISCONSIN ALUMNI RESEARCH FOUNDATION (US) 1998-05-22 WO disclosed
US-5700659-A GENETIC ENGINEERED GENE FOR GENE EXPRESSION KABUSHIKI KAISHA TOYOTA CHUO KENKUSHO (JP) 1997-12-23 US disclosed
EP-0749493-A1 INHIBITION OF PROTEASE ACTIVITY OF HUMAN WHOLE BLOOD CELL LYSATES Ciba Corning Diagnostics Corp. (US) 1996-12-27 EP disclosed
EP-0720657-A1 BIOLOGICALLY RELEVANT METHODS FOR THE RAPID DETERMINATION OF STERILITY NORTH AMERICAN SCIENCE ASSOCIATES INCORPORATED (US) 1996-07-10 EP disclosed
US-5496719-A THERMOSTABILITY, CATALYST FOR DISULFIDE EXCHANGE IN PROTEINS KABUSHIKI KAISHA TOYOTA CHUO KENKYUSHO (JP) 1996-03-05 US disclosed
US-5486459-A Biologically relevant methods for the rapid determination of sterility MEDICAL COLLEGE OF OHIO (US) 1996-01-23 US disclosed
WO-1995035366-A1 ANIMAL MODEL FOR ALZHEIMER'S DISEASE THE TRUSTEES OF THE UNIVERSITY OF PENNSYLVANIA (US) 1995-12-28 WO disclosed
WO-1995024500-A1 INHIBITION OF PROTEASE ACTIVITY OF HUMAN WHOLE BLOOD CELL LYSATES CIBA CORNING DIAGNOSTICS CORP. (US) 1995-09-14 WO disclosed
WO-1995008639-A1 BIOLOGICALLY RELEVANT METHODS FOR THE RAPID DETERMINATION OF STERILITY NORTH AMERICAN SCIENCE ASSOCIATES, INC. (US) 1995-03-30 WO disclosed
WO-1994012640-A1 RECOMBINANT NUCLEIC ACID, POLYPEPTIDE MATERIAL CODED THEREBY AND TRANSMISSION BLOCKING VACCINE BASED THEREON FOR CONTROLLING THE MALARIA PARASITE $i(PLASMODIUM FALCIPARUM ) STICHTING KATHOLIEKE UNIVERSITEIT (NL) 1994-06-09 WO disclosed
US-5310880-A Chromatography, alkali halide, acid solution THE GENERAL HOSPITAL CORPORATION (US) 1994-05-10 US disclosed
EP-0554064-A1 Vaccine against schistosomiasis YEDA RESEARCH AND DEVELOPMENT CO. LTD. (IL) 1993-08-04 EP disclosed
WO-1992018145-A1 PURIFICATION OF MÜLLERIAN INHIBITING SUBSTANCE THE GENERAL HOSPITAL CORPORATION (US) 1992-10-29 WO disclosed
EP-0323802-A2 Monoclonal antibodies against, and cell surface antigen of, lung carcinoma SANDOZ AG (CH) 1989-07-12 EP disclosed
US-4677069-A Clam derived proteinases CORNELL RESEARCH FOUNDATION, INC. (US) 1987-06-30 US disclosed
US-4677069-A Clam derived proteinases CORNELL RESEARCH FOUNDATION, INC. (US) 1987-06-30 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (10 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20140349969-A1 COMPOUNDS AND METHODS FOR TREATING PAIN TRPV1, ACHE, OPRL1 MMP9 664/4885MMP2 882/4885ITGB3 1250/4885
US-12551475-B2 Methods and compositions for treating RNA viral infections SARS1, EIF2AK2, SNRPE MMP9 2494/4885MMP2 4687/4885ITGB3 2892/4885
US-20070077283-A1 METHOD OF ENHANCING TRANSMUCOSAL DELIVERY OF THERAPEUTIC COMPOUNDS PGF, PLAT, PTAFR MMP9 279/4885MMP2 255/4885ITGB3 680/4885
US-20130252924-A1 Compounds and Methods for Treating Pain TRPV1, ACHE, OPRL1 MMP9 664/4885MMP2 882/4885ITGB3 1250/4885
US-20020058288-A1 Compound for use in the detection and prevention of parasitic infection of humans CD4, OGA, GPI MMP9 3744/4885MMP2 1576/4885ITGB3 261/4885
US-20250025454-A1 USE OF PIPENDOXIFENE TO TREAT SARS-COV-2 INFECTION EIF2AK2, ACE2, SARS1 MMP9 2057/4885MMP2 3595/4885ITGB3 3439/4885
US-20190216779-A1 USE OF NEUROKININ-1 ANTAGONISTS TO TREAT A VARIETY OF PRURITIC CONDITIONS BDKRB2, BDKRB1, PBK MMP9 2951/4885MMP2 3262/4885ITGB3 2318/4885
US-20180235931-A1 USE OF NEUROKININ-1 ANTAGONISTS AS ANTITUSSIVES OPRK1, TAC3, BRS3 MMP9 4261/4885MMP2 2923/4885ITGB3 1824/4885
US-20090054326-A1 FORMULATIONS FOR ENHANCED MUCOSAL DELIVERY OF PYY NPY1R, NPY5R, NPY2R MMP9 2387/4885MMP2 2339/4885ITGB3 4332/4885
US-20230346792-A1 COMPOSITIONS AND METHODS FOR TREATING LUNG INFLAMMATION ACE2, TMPRSS2, VIPR1 MMP9 402/4885MMP2 1445/4885ITGB3 2173/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.