SCHEMBL7965454

SCHEMBL7965454

OC(CCN1CCC(O)(c2cncc3ccccc23)CC1)Oc1ccc2ccccc2c1

nearest known ligand 0.36

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
OPRL1 P41146 3/20 0.36
KDM4E B2RXH2 2/20 0.36
KMT2A Q03164 2/20 0.36
MEN1 O00255 1/20 0.36
CCR1 P32246 3/20 0.35
SLC6A1 P30531 2/20 0.34
SLC6A12 P48065 2/20 0.34
SLC6A11 P48066 2/20 0.34
SLC6A13 Q9NSD5 1/20 0.34
HRH3 Q9Y5N1 2/20 0.34
HRH1 P35367 1/20 0.34
HTR1A P08908 2/20 0.33
DRD3 P35462 1/20 0.33
CYP3A4 P08684 1/20 0.33
CYP2C9 P11712 1/20 0.33
CYP2C19 P33261 1/20 0.33
OPRM1 P35372 1/20 0.33
TACR2 P21452 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7967096 0.90 TUBB4A (0.38) OPRL1SLC6A1SLC6A12SLC6A11SLC6A13
SCHEMBL8139378 0.87 SLC6A1 (0.34) OPRL1KDM4EKMT2AMEN1CCR1
SCHEMBL7962999 0.87 OPRL1 (0.40) OPRL1CCR1HTR1AOPRM1
SCHEMBL7963100 0.87 SLC6A1 (0.34) OPRL1KDM4EKMT2AMEN1CCR1
SCHEMBL7965451 0.80 SMN1; SMN2 (0.55) KDM4EKMT2AMEN1HTR1ACYP3A4
SCHEMBL7965345 0.80 SLC6A1 (0.34) OPRL1SLC6A1SLC6A12SLC6A11SLC6A13
SCHEMBL7965744 0.79 HTR1A (0.36) SLC6A1SLC6A12SLC6A11SLC6A13HTR1A
SCHEMBL7967126 0.79 ABCB1 (0.39) DRD3
SCHEMBL7200725 0.78 OPRL1 (0.41) OPRL1KDM4EKMT2AMEN1CCR1
SCHEMBL7965447 0.78 HRH3 (0.36) KDM4EHRH3HRH1DRD3CYP3A4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6242450-B1 SUBSTITUTED PIPERIDINES ELI LILLY AND COMPANY 2001-06-05 US disclosed
WO-2000006166-A1 5-HT1F ANTAGONISTS ELI LILLY AND COMPANY (US) 2000-02-10 WO disclosed
EP-0976746-A1 5-HT1F antagonists ELI LILLY AND COMPANY (US) 2000-02-02 EP disclosed