SCHEMBL7967019

SCHEMBL7967019

COc1cc(C(=O)N(C)c2ccc(C)cc2OCCCCC(=C=O)N2CCN(C)CC2)ccc1NC(=O)c1ccc2c(c1)N(C(=O)OC(C)(C)C)CC2

nearest known ligand 0.48

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
CPT1A P50416 3/20 0.34
CPT1B Q92523 3/20 0.34
ADRA1D P25100 5/20 0.33
ADRA1A P35348 5/20 0.33
ADRA1B P35368 5/20 0.33
AVPR2 P30518 2/20 0.33
AVPR1A P37288 2/20 0.33
AVPR1B P47901 2/20 0.33
CHRM4 P08173 1/20 0.33
DRD2 P14416 1/20 0.33
HTR7 P34969 1/20 0.33
CPT2 P23786 2/20 0.32
TP53 P04637 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7967020 0.93 AVPR2 (0.38) CPT1ACPT1BADRA1DADRA1AADRA1B
SCHEMBL7969562 0.87 MAPK11 (0.36) CPT1ACPT1BADRA1DADRA1AADRA1B
SCHEMBL7971950 0.83 AVPR2 (0.41) ADRA1DADRA1AADRA1BAVPR2AVPR1A
SCHEMBL7475346 0.83 MAP3K7 (0.32) ADRA1DADRA1AADRA1BAVPR2AVPR1A
SCHEMBL7474244 0.83 AVPR2 (0.33) ADRA1DADRA1AADRA1BAVPR2AVPR1A
Hydrochloric Acid SCHEMBL7476852 0.82 MAPK11 (0.36) ADRA1DADRA1AADRA1B
SCHEMBL7955154 0.81 ADRA1D (0.32) ADRA1DADRA1AADRA1BAVPR2AVPR1A
SCHEMBL7478471 0.80 MAP3K7 (0.36) ADRA1DADRA1AADRA1BAVPR2AVPR1A
SCHEMBL7475173 0.80 AVPR2 (0.32) AVPR2AVPR1AAVPR1B
SCHEMBL7342048 0.79 LMNA (0.38) TP53

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6316482-B1 FOR THERAPY AND PROPHYLAXIS OF HYPERTENSION, HEART FAILURE, RENAL INSUFFICIENCY, EDEMA, ASCITES, VASOPRESSIN PARASECRETION SYNDROME, HEPATOCIRRHOSIS, HYPONATREMIA, HYPOKALEMIA, DIABETIC, CIRCULATION DISORDER, CEREBROVASCULAR DISEASE FUJISAWA PHARMACEUTICAL CO., LTD. (JP) 2001-11-13 US disclosed