SCHEMBL7969815

SCHEMBL7969815

COC(=O)C1=Cc2cc(-c3cc(C)cs3)ccc2S(=O)(=O)CC1

nearest known ligand 0.36

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
HDAC1 Q13547 4/20 0.36
HDAC2 Q92769 4/20 0.36
HDAC3 O15379 3/20 0.36
HSD17B10 Q99714 2/20 0.36
ALDH1A1 P00352 1/20 0.36
MAPT P10636 1/20 0.36
TSHR P16473 1/20 0.36
MAPK1 P28482 1/20 0.36
TNFRSF1A P19438 3/20 0.35
CA12 O43570 4/20 0.33
CA9 Q16790 4/20 0.33
ABL1 P00519 1/20 0.33
SLC6A7 Q99884 1/20 0.32
CYP46A1 Q9Y6A2 1/20 0.32
CA2 P00918 1/20 0.31
PRKCZ Q05513 1/20 0.31
LMNA P02545 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7975481 0.88 HDAC1 (0.36) HDAC1HDAC2HDAC3TNFRSF1AABL1
SCHEMBL7975083 0.84 CA12 (0.39) HSD17B10ALDH1A1MAPTTSHRMAPK1
SCHEMBL7931191 0.84 HDAC1 (0.35) HDAC1HDAC2HDAC3ALDH1A1TNFRSF1A
SCHEMBL7931232 0.81 HDAC2 (0.35) HDAC1HDAC2HDAC3MAPTTSHR
SCHEMBL7934057 0.80 SLC6A3 (0.40) ALDH1A1MAPTCA12CA9LMNA
SCHEMBL7969052 0.79 CA12 (0.42) ALDH1A1MAPK1CA12CA9CA2
SCHEMBL7934163 0.79 KDM4E (0.45) ALDH1A1MAPTCA12CA9CA2
SCHEMBL7969353 0.79 SLC6A3 (0.40) ALDH1A1MAPTCA12CA9CA2
SCHEMBL7969661 0.78 PTGDR2 (0.41) CA12CA9CA2LMNA
SCHEMBL7922070 0.78 L3MBTL1 (0.35) ALDH1A1MAPTTSHRCA12CA9

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6235771-B1 AIDS THERPAY TAKEDA CHEMICAL INDUSTRIES, LTD. (JP) 2001-05-22 US disclosed