SCHEMBL7971104

SCHEMBL7971104

COC1=C(OC)C(=O)C2=C(CC(CCCCCCCC(N)=O)(C(N)=O)C2)C1=O

nearest known ligand 0.36

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
APEX1 P27695 3/20 0.36
CYP4F2 P78329 1/20 0.31
CYP4A11 Q02928 1/20 0.31
LMNA P02545 1/20 0.30
PGR P06401 1/20 0.30
CYP3A4 P08684 1/20 0.30
CYP2D6 P10635 1/20 0.30
MAPT P10636 1/20 0.30
CYP2C9 P11712 1/20 0.30
MAOA P21397 1/20 0.30
TBXA2R P21731 1/20 0.30
MAPK1 P28482 1/20 0.30
AVPR2 P30518 1/20 0.30
CYP2C19 P33261 1/20 0.30
HTR2B P41595 1/20 0.30
HTT P42858 1/20 0.30
PDE3A Q14432 1/20 0.30
SIRT2 Q8IXJ6 1/20 0.30
SLC29A1 Q99808 1/20 0.30
TDP1 Q9NUW8 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7971265 0.81 ALDH1A1 (0.37) APEX1LMNAPDE3ATDP1
SCHEMBL7961097 0.77 CYP4F2 (0.32) CYP4F2CYP4A11
SCHEMBL7977541 0.76 CYP4F2 (0.35) APEX1CYP4F2CYP4A11CYP3A4TDP1
SCHEMBL7974475 0.73 CYP4F2 (0.43) APEX1CYP4F2CYP4A11LMNAPGR
SCHEMBL7974447 0.72 CYP4F2 (0.43) CYP4F2CYP4A11LMNAPGRCYP3A4
SCHEMBL2356683 0.72 MME (0.37) LMNAMAPTTDP1
SCHEMBL1165196 0.71 KDM4E (0.31) CYP3A4CYP2C19
SCHEMBL5613217 0.71 KDM4E (0.31) CYP3A4CYP2C19
SCHEMBL11787061 0.71 KDM4E (0.31) CYP3A4CYP2C19
SCHEMBL675034 0.70 TBXAS1 (0.33)

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6326369-B1 ALZHEIMER'S DISEASE TAKEDA CHEMICALS INDUSTRIES, LTD. (JP) 2001-12-04 US disclosed
EP-0968164-A1 BICYCLIC QUINONE COMPOUNDS, THEIR PRODUCTION AND USE Takeda Chemical Industries, Ltd. (JP) 2000-01-05 EP disclosed
WO-1998033758-A1 BICYCLIC QUINONE COMPOUNDS, THEIR PRODUCTION AND USE TAKEDA CHEMICAL INDUSTRIES, LTD. (JP) 1998-08-06 WO disclosed