SCHEMBL7971509

SCHEMBL7971509

COc1c2c(c(OC)c(OC)c1OC)CC(CCCCCCCCN1CCN(C(c3ccccc3)c3ccccc3)CC1)C2

nearest known ligand 0.54

Predicted protein targets (top 9)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 1/20 0.51
L3MBTL1 Q9Y468 1/20 0.51
MEN1 O00255 1/20 0.50
KMT2A Q03164 1/20 0.50
P2RX7 Q99572 6/20 0.48
ALOX5 P09917 6/20 0.48
DRD2 P14416 1/20 0.47
DRD3 P35462 1/20 0.47
ADRA1B P35368 1/20 0.45

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7971522 0.83 CCR3 (0.50)
Hydrochloric Acid SCHEMBL7974723 0.82 CCR3 (0.49)
Hydrochloric Acid SCHEMBL7977428 0.79 SIGMAR1 (0.52) MEN1KMT2ADRD2
SCHEMBL7971195 0.76 KCNH2 (0.56) DRD2DRD3ADRA1B
SCHEMBL7977198 0.74 ALDH1A1 (0.43) ALDH1A1KMT2A
SCHEMBL7961134 0.71 HCAR2 (0.31)
SCHEMBL6617019 0.71 DRD2 (0.62) MEN1KMT2AP2RX7DRD2DRD3
SCHEMBL7383823 0.71 DRD2 (0.66) ALDH1A1L3MBTL1P2RX7DRD2DRD3
SCHEMBL11938950 0.71 OPRM1 (0.68) P2RX7DRD2DRD3ADRA1B
SCHEMBL7974371 0.71 HTR1A (0.48) ALDH1A1L3MBTL1MEN1KMT2ADRD2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6326369-B1 ALZHEIMER'S DISEASE TAKEDA CHEMICALS INDUSTRIES, LTD. (JP) 2001-12-04 US disclosed
EP-0968164-A1 BICYCLIC QUINONE COMPOUNDS, THEIR PRODUCTION AND USE Takeda Chemical Industries, Ltd. (JP) 2000-01-05 EP disclosed
WO-1998033758-A1 BICYCLIC QUINONE COMPOUNDS, THEIR PRODUCTION AND USE TAKEDA CHEMICAL INDUSTRIES, LTD. (JP) 1998-08-06 WO disclosed