SCHEMBL7972575

SCHEMBL7972575

COC[C@@H]1OC(=O)N(C(=O)Oc2ccc([N+](=O)[O-])cc2)[C@H]1c1ccc(F)c(F)c1

nearest known ligand 0.40

Predicted protein targets (top 8)

geneUniProtsupporting neighboursconfidence
MGLL Q99685 2/20 0.39
BCL9 O00512 1/20 0.35
CTNNB1 P35222 1/20 0.35
KDM1A O60341 1/20 0.35
GAA P10253 1/20 0.34
CYP1A2 P05177 1/20 0.34
CYP2D6 P10635 1/20 0.34
FAAH O00519 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5662288 0.86 ADRA1A (0.42) MGLLBCL9CTNNB1KDM1AGAA
SCHEMBL8174001 0.86 ADRA1A (0.42) MGLLBCL9CTNNB1KDM1AGAA
SCHEMBL5658840 0.86 ADRA1A (0.42) MGLLBCL9CTNNB1KDM1AGAA
SCHEMBL7747876 0.84 MGLL (0.39) MGLLKDM1AGAA
SCHEMBL7747880 0.84 MGLL (0.39) MGLLKDM1AGAA
SCHEMBL7995847 0.84 MGLL (0.39) MGLLKDM1AGAA
SCHEMBL6953243 0.84 MGLL (0.38) MGLLCYP1A2CYP2D6FAAH
SCHEMBL7966161 0.81 MGLL (0.43) MGLLCYP1A2CYP2D6FAAH
SCHEMBL8173301 0.81 MGLL (0.43) MGLLCYP1A2CYP2D6FAAH
SCHEMBL7972617 0.79 ADRA1A (0.39)

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6228870-B1 BENIGN PROSTATIC HYPERPLASIA; REDUCTION OF HYPOTENSION SIDE EFFECT MERCK & CO., INC. 2001-05-08 US disclosed