SCHEMBL7976201

SCHEMBL7976201

C=CCCCN(C)C(=O)[C@H](Cc1c[nH]c2ccccc12)NC(=O)O

nearest known ligand 0.59

Predicted protein targets (top 10)

geneUniProtsupporting neighboursconfidence
TACR1 P25103 2/20 0.59
MMP9 P14780 1/20 0.54
MMP8 P22894 1/20 0.54
MMP14 P50281 1/20 0.54
ALOX15 P16050 1/20 0.52
CCKBR P32239 6/20 0.51
ITGB2 P05107 1/20 0.49
ICAM1 P05362 1/20 0.49
ITGAL P20701 1/20 0.49
ACE P12821 3/20 0.48

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7976198 1.00 TACR1 (0.59) TACR1MMP9MMP8MMP14ALOX15
SCHEMBL7993694 0.87 MMP2 (0.54) TACR1MMP9MMP8MMP14ACE
SCHEMBL7989362 0.84 KDM4E (0.55) TACR1MMP9MMP8MMP14
SCHEMBL7989539 0.83 MMP9 (0.52) TACR1MMP9MMP8MMP14CCKBR
SCHEMBL7989529 0.83 MMP9 (0.52) TACR1MMP9MMP8MMP14CCKBR
SCHEMBL3780103 0.82 MMP9 (0.77) TACR1MMP9MMP8MMP14ALOX15
SCHEMBL8200364 0.81 TACR1 (0.86) TACR1MMP9MMP8MMP14ALOX15
SCHEMBL8200367 0.81 TACR1 (0.86) TACR1MMP9MMP8MMP14ALOX15
SCHEMBL17870487 0.79 NMBR (0.58) TACR1ALOX15
SCHEMBL17870489 0.79 NMBR (0.58) TACR1ALOX15

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2001040198-A2 MACROCYCLIC HYDROXAMIC ACID DERIVATIVES AND THEIR USE AS ANTIMICROBIAL AGENTS AVENTIS PHARMA S.A. (FR) 2001-06-07 WO disclosed