SCHEMBL7976947

SCHEMBL7976947

CC(C)(COc1ccc(C(O)c2ccc(OC(F)F)c(OC(F)F)c2)cn1)c1ccc(F)cc1

nearest known ligand 0.39

Predicted protein targets (top 7)

geneUniProtsupporting neighboursconfidence
PDE4A P27815 19/20 0.39
KCNH2 Q12809 3/20 0.39
PDE4D Q08499 1/20 0.35
CYP2C9 P11712 1/20 0.34
CYP2C19 P33261 1/20 0.34
EPHX2 P34913 1/20 0.34
CYP2J2 P51589 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7991436 0.88 PDE4A (0.38) PDE4AKCNH2PDE4D
SCHEMBL7978041 0.82 PDE4A (0.53) PDE4AKCNH2
SCHEMBL7991279 0.80 PDE4A (0.33) PDE4AKCNH2PDE4DCYP2C9CYP2C19
SCHEMBL7383406 0.80 PDE4A (0.65) PDE4AKCNH2
SCHEMBL7991120 0.72 ALOX5 (0.39) PDE4AKCNH2
SCHEMBL7991049 0.71 PDE4A (0.41) PDE4AKCNH2
SCHEMBL7989179 0.70 PDE4A (0.37) PDE4AKCNH2
SCHEMBL7367599 0.70 PDE4A (0.43) PDE4AKCNH2
SCHEMBL7977119 0.69 PDE4A (0.54) PDE4AKCNH2
SCHEMBL7990920 0.69 THRB (0.35) CYP2C9CYP2C19EPHX2CYP2J2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6180650-B1 ANTIINFLAMMATORY AGENTS; RESPIRATORY SYSTEM DISORDERS; SKIN DISORDERS; ANTITUMOR AGENTS MERCK FROSST CANADA & CO. (CA) 2001-01-30 US disclosed