SCHEMBL7991279

SCHEMBL7991279

CCOC(=O)C(c1ccncc1)C(c1ccc(OCC(C)(C)c2ccc(F)cc2)nc1)c1ccc(OC(F)F)c(OC(F)F)c1

nearest known ligand 0.33

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
PDE4A P27815 14/20 0.33
KCNH2 Q12809 2/20 0.33
FBP1 P09467 1/20 0.31
CYP2C9 P11712 1/20 0.31
CYP2C19 P33261 1/20 0.31
EPHX2 P34913 1/20 0.31
CYP2J2 P51589 1/20 0.31
PDE4B Q07343 2/20 0.31
PDE4C Q08493 2/20 0.31
PDE4D Q08499 2/20 0.31
MAPK14 Q16539 2/20 0.31
CXCR1 P25024 1/20 0.30
CXCR2 P25025 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7976947 0.80 PDE4A (0.39) PDE4AKCNH2CYP2C9CYP2C19EPHX2
SCHEMBL7908336 0.80 PDE4A (0.38) PDE4AKCNH2FBP1PDE4BPDE4C
SCHEMBL7991148 0.79 PDE4A (0.34) PDE4AFBP1PDE4BPDE4CPDE4D
SCHEMBL7978041 0.79 PDE4A (0.53) PDE4AKCNH2
SCHEMBL7992704 0.78 F7 (0.36) PDE4AKCNH2PDE4BPDE4CPDE4D
SCHEMBL7996011 0.77 LMNA (0.41) PDE4APDE4BPDE4CPDE4D
SCHEMBL7991436 0.77 PDE4A (0.38) PDE4AKCNH2PDE4D
SCHEMBL7990957 0.77 RAB9A (0.39) PDE4AFBP1PDE4BPDE4CPDE4D
SCHEMBL7994826 0.75 PDE4B (0.33) PDE4AFBP1PDE4BPDE4CPDE4D
SCHEMBL7904298 0.72 PDE4A (0.43) PDE4APDE4BPDE4CPDE4D

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6180650-B1 ANTIINFLAMMATORY AGENTS; RESPIRATORY SYSTEM DISORDERS; SKIN DISORDERS; ANTITUMOR AGENTS MERCK FROSST CANADA & CO. (CA) 2001-01-30 US disclosed