SCHEMBL7991049

SCHEMBL7991049

CS(=O)(=O)c1ccc(COc2ccc(C(O)c3ccc(OC(F)F)c(OC(F)F)c3)cn2)cc1

nearest known ligand 0.41

Predicted protein targets (top 6)

geneUniProtsupporting neighboursconfidence
PDE4A P27815 18/20 0.41
KCNH2 Q12809 2/20 0.41
GPR119 Q8TDV5 1/20 0.40
ADRB2 P07550 1/20 0.36
ADRB1 P08588 1/20 0.36
ADRB3 P13945 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7994656 0.88 PDE4A (0.39) PDE4AKCNH2GPR119
SCHEMBL7991120 0.84 ALOX5 (0.39) PDE4AKCNH2
SCHEMBL7990922 0.83 PDE4A (0.53) PDE4AKCNH2
SCHEMBL7462478 0.82 PDE4A (0.64) PDE4AKCNH2
SCHEMBL7992704 0.81 F7 (0.36) PDE4AKCNH2GPR119
SCHEMBL7976947 0.71 PDE4A (0.39) PDE4AKCNH2
SCHEMBL7991261 0.69 HSPB1 (0.48) PDE4A
SCHEMBL7367599 0.69 PDE4A (0.43) PDE4AKCNH2
SCHEMBL7977065 0.69 LMNA (0.51) PDE4A
SCHEMBL7380926 0.68 PDE4A (0.76) PDE4AKCNH2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6180650-B1 ANTIINFLAMMATORY AGENTS; RESPIRATORY SYSTEM DISORDERS; SKIN DISORDERS; ANTITUMOR AGENTS MERCK FROSST CANADA & CO. (CA) 2001-01-30 US disclosed