SCHEMBL7984773

SCHEMBL7984773

Cc1c(O)cc2c(c1C)C(=O)c1nc3nonc3nc1-2

nearest known ligand 0.41

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
PTGES O14684 3/20 0.41
USP8 P40818 1/20 0.33
USP7 Q93009 1/20 0.33
MEN1 O00255 1/20 0.31
LMNA P02545 1/20 0.31
TP53 P04637 1/20 0.31
MAPK1 P28482 1/20 0.31
HTT P42858 1/20 0.31
KMT2A Q03164 1/20 0.31
TDP1 Q9NUW8 1/20 0.31
L3MBTL1 Q9Y468 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7994928 0.80 PTGES (0.42) PTGESUSP8USP7MEN1LMNA
SCHEMBL7983849 0.73 PTGES (0.57) PTGESUSP8MEN1LMNATP53
SCHEMBL7984866 0.72 PTGES (0.39) PTGESMEN1LMNAKMT2AL3MBTL1
SCHEMBL7984632 0.70 USP8 (0.60) PTGESUSP8USP7MEN1LMNA
SCHEMBL7998365 0.68 USP7 (0.59) PTGESUSP8USP7MEN1LMNA
SCHEMBL7996719 0.64 PTGES (0.64) PTGESUSP8USP7MEN1LMNA
SCHEMBL7996577 0.62 PTGES (0.49) PTGESUSP8USP7MEN1LMNA
SCHEMBL7984622 0.62 PTGES (0.52) PTGESUSP8USP7MEN1LMNA
SCHEMBL31696139 0.62 USP7 (0.59) PTGESUSP8USP7MEN1LMNA
SCHEMBL31696105 0.62 PTGES (0.52) PTGESUSP8USP7MEN1LMNA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2001079209-A2 DIAZAFLUORENONE IL-8 ANTAGONISTS MILLENNIUM PHARMACEUTICALS, INC. (US) 2001-10-25 WO claimed
WO-2001079209-A2 DIAZAFLUORENONE IL-8 ANTAGONISTS MILLENNIUM PHARMACEUTICALS, INC. (US) 2001-10-25 WO disclosed