SCHEMBL7988652

SCHEMBL7988652

NC(=O)c1cccc(N(S(=O)(=O)/C=C/c2ccccc2)S(=O)(=O)/C=C/c2ccccc2)c1

nearest known ligand 0.44

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PPARG P37231 1/20 0.44
PTGS2 P35354 4/20 0.40
PTGS1 P23219 3/20 0.40
HTR2A P28223 1/20 0.40
HTR2C P28335 1/20 0.40
PARP1 P09874 6/20 0.40
MAPT P10636 2/20 0.40
RECQL P46063 2/20 0.40
POLB P06746 1/20 0.40
CYP3A4 P08684 1/20 0.40
TSHR P16473 1/20 0.40
CYP2C19 P33261 1/20 0.40
BLM P54132 1/20 0.40
PMP22 Q01453 1/20 0.40
HSD17B10 Q99714 1/20 0.40
TDP1 Q9NUW8 1/20 0.40
L3MBTL1 Q9Y468 1/20 0.40
CRY1 Q16526 1/20 0.38
CRY2 Q49AN0 1/20 0.38
KMT2A Q03164 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8000279 0.85 KMT2A (0.43) PPARGHTR2AHTR2CPARP1MAPT
SCHEMBL7988658 0.83 PPARG (0.44) PPARGMAPTPOLBTSHRCYP2C19
SCHEMBL8001632 0.77 MAPT (0.48) PPARGMAPTLMNAMAOB
SCHEMBL7988653 0.77 MAOB (0.41) PPARGMAPTKMT2ALMNAMAOB
SCHEMBL8004163 0.75 TSHR (0.42) PPARGMAPTPOLBTSHRCYP2C19
SCHEMBL28179497 0.74 TTR (0.59) PARP1MAPTRECQLPOLBCYP3A4
SCHEMBL8002290 0.74 MAOB (0.47) MAPTKMT2AMAOB
SCHEMBL8001633 0.74 NFE2L2 (0.50) PPARGMAPTCYP3A4HSD17B10KMT2A
SCHEMBL7998748 0.74 CYP19A1 (0.41) PPARGMAPTPOLBKMT2ALMNA
SCHEMBL7988661 0.70 PPARG (0.49) PPARGMAPTTSHRL3MBTL1KMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2009120783-A1 HIGH AFFINITY INHIBITORS OF HEPATITIS C VIRUS NS3/4A PROTEASE THE JOHNS HOPKINS UNIVERSITY (US) 2009-10-01 WO disclosed