SCHEMBL7990975

SCHEMBL7990975

COc1ccccc1CNc1nc(=O)cc(-c2ccncc2)[nH]1

nearest known ligand 0.49

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HSD17B10 Q99714 3/20 0.49
KDM1A O60341 1/20 0.49
GAA P10253 1/20 0.49
RCOR1 Q9UKL0 1/20 0.49
PDE9A O76083 4/20 0.48
KMT2A Q03164 2/20 0.47
MEN1 O00255 1/20 0.47
ALDH1A1 P00352 1/20 0.45
CYP1A2 P05177 3/20 0.44
CYP3A4 P08684 3/20 0.44
CYP2D6 P10635 3/20 0.44
CYP2C19 P33261 3/20 0.44
TSHR P16473 2/20 0.44
CLK4 Q9HAZ1 2/20 0.44
ROCK2 O75116 2/20 0.44
ROCK1 Q13464 1/20 0.44
PRKCA P17252 1/20 0.44
GRK2 P25098 1/20 0.44
ABL1 P00519 1/20 0.43
SRC P12931 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7989732 0.82 GAA (0.52) HSD17B10GAAKMT2AMEN1ALDH1A1
SCHEMBL5380552 0.80 XDH (0.53) HSD17B10KMT2AMEN1ALDH1A1CLK4
SCHEMBL7992854 0.73 GPR84 (0.41) KMT2AMEN1ROCK2ROCK1PRKCA
SCHEMBL3830998 0.73 MEN1 (0.54) PDE9AKMT2AMEN1ALDH1A1ROCK2
SCHEMBL7989847 0.73 CDC7 (0.43) CLK4ROCK2ROCK1PRKCAGRK2
SCHEMBL7996288 0.72 MTNR1A (0.46) CYP3A4CYP2D6CLK4ROCK2ROCK1
SCHEMBL7996305 0.72 CDC7 (0.45) KMT2AMEN1ALDH1A1CDC7
SCHEMBL7993806 0.72 FABP1 (0.45) GAATSHRCLK4ROCK2PRKCA
SCHEMBL7991079 0.72 ALOX5 (0.41) HSD17B10KMT2AMEN1ALDH1A1CLK4
SCHEMBL5375269 0.71 CDC7 (0.43) CDC7

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2001070727-A1 2-(ARYLALKYLAMINO)PYRIMIDONE DERIVATIVES AND 2-(HETEROARYLALKYLAMINO)PYRIMIDONE DERIVATIVES SANOFI-SYNTHELABO (FR) 2001-09-27 WO claimed