SCHEMBL7994539

SCHEMBL7994539

COc1ccc2c(C)cn(CC(C)(N)OC(=O)/C=C\C(=O)OC(C)(N)Cn3cc(C)c4ccc(OC)cc43)c2c1

nearest known ligand 0.38

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 1/20 0.38
PDE4A P27815 2/20 0.38
PDE4B Q07343 2/20 0.38
PDE4C Q08493 2/20 0.38
PDE4D Q08499 2/20 0.38
MEN1 O00255 1/20 0.38
KMT2A Q03164 1/20 0.38
HDAC1 Q13547 2/20 0.37
HDAC2 Q92769 2/20 0.37
HDAC6 Q9UBN7 2/20 0.37
ESR1 P03372 1/20 0.37
CNR1 P21554 3/20 0.36
CNR2 P34972 2/20 0.36
PLA2G2A P14555 3/20 0.35
DYRK1A Q13627 2/20 0.35
SLC22A12 Q96S37 1/20 0.34
PLA2G10 O15496 1/20 0.34
HTR6 P50406 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6364121 0.79 SLC22A12 (0.39) ALDH1A1KMT2AESR1DYRK1ASLC22A12
SCHEMBL8959747 0.79 AR (0.44) ALDH1A1
SCHEMBL8959949 0.77 SLC22A12 (0.35) PDE4APDE4BPDE4CPDE4DKMT2A
SCHEMBL8959667 0.73 TRPM5 (0.38) PLA2G2A
SCHEMBL8959711 0.72 HTR2C (0.45) ALDH1A1MEN1KMT2A
Fumaric Acid SCHEMBL7994542 0.72 HTR2C (0.46) PDE4APDE4BPDE4CPDE4DMEN1
Maleic Acid SCHEMBL7994532 0.72 HTR2C (0.46) PDE4APDE4BPDE4CPDE4DMEN1
SCHEMBL7850213 0.71 HTR6 (0.49) ALDH1A1PDE4APDE4BPDE4CPDE4D
SCHEMBL8959547 0.70 HTR2C (0.45) HDAC1HDAC2HDAC6
SCHEMBL27342171 0.70 HTR2C (0.45) HDAC1HDAC2HDAC6

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2001040183-A1 1-AMINOALKYL-1H-INDOLES FOR TREATING GLAUCOMA ALCON UNIVERSAL LTD. (CH) 2001-06-07 WO disclosed