SCHEMBL7997110

SCHEMBL7997110

CCN(C(=O)CNS(=O)(=O)Cc1ccccc1Cl)[C@@H]1CN(C(=O)[C@@H](NC(=O)c2cc3ccccc3[nH]2)C(C)(C)C)C1C

nearest known ligand 0.38

Predicted protein targets (top 10)

geneUniProtsupporting neighboursconfidence
DRD2 P14416 8/20 0.38
CYP51A1 Q16850 2/20 0.37
PYGL P06737 3/20 0.37
STAT6 P42226 1/20 0.34
CCKBR P32239 4/20 0.34
DRD3 P35462 7/20 0.34
HTR1A P08908 4/20 0.34
HTR2A P28223 4/20 0.34
HTR2C P28335 4/20 0.34
DRD4 P21917 2/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8005363 0.87 PYGL (0.41) DRD2CYP51A1PYGLDRD3
SCHEMBL7995570 0.84 DRD2 (0.38) DRD2CYP51A1PYGLSTAT6CCKBR
SCHEMBL8004708 0.84 PYGL (0.39) DRD2CYP51A1PYGLSTAT6DRD3
SCHEMBL4049377 0.82 CYP51A1 (0.39) DRD2CYP51A1PYGLSTAT6CCKBR
SCHEMBL8008794 0.81 STAT6 (0.40) DRD2CYP51A1PYGLSTAT6CCKBR
SCHEMBL8008195 0.77 TRPV4 (0.43) DRD2CYP51A1PYGLCCKBR
SCHEMBL8007233 0.77 DRD2 (0.37) DRD2CYP51A1PYGLSTAT6CCKBR
SCHEMBL7995203 0.77 DRD2 (0.37) DRD2CYP51A1PYGLSTAT6CCKBR
SCHEMBL8008199 0.75 DRD2 (0.44) DRD2CYP51A1PYGLSTAT6CCKBR
SCHEMBL8010535 0.75 DRD2 (0.37) DRD2CYP51A1PYGLSTAT6CCKBR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2009111680-A1 TRPV4 ANTAGONISTS SMITHLINE BEECHAM CORPORATION (US) 2009-09-11 WO disclosed