SCHEMBL4049377

SCHEMBL4049377

CC(C)(C)[C@H](NC(=O)c1cc2ccccc2[nH]1)C(=O)N1C[C@@H]2C[C@H]1CN2C(=O)CNS(=O)(=O)Cc1ccccc1Cl

nearest known ligand 0.39

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
CYP51A1 Q16850 2/20 0.39
DRD2 P14416 9/20 0.39
PYGL P06737 1/20 0.36
STAT6 P42226 1/20 0.35
DRD3 P35462 8/20 0.35
DRD4 P21917 5/20 0.35
HTR1A P08908 4/20 0.35
HTR2A P28223 4/20 0.35
HTR2C P28335 4/20 0.35
TAS1R3 Q7RTX0 1/20 0.35
TAS1R1 Q7RTX1 1/20 0.35
CCKBR P32239 1/20 0.34
KCNH2 Q12809 1/20 0.34
DRD1 P21728 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4057673 0.86 PYGL (0.39) CYP51A1DRD2PYGLSTAT6DRD3
SCHEMBL4057362 0.86 PYGL (0.39) CYP51A1DRD2PYGLDRD3
SCHEMBL4050168 0.84 DRD2 (0.36) CYP51A1DRD2PYGLSTAT6DRD3
SCHEMBL19856906 0.83 DRD2 (0.45) CYP51A1DRD2PYGLSTAT6DRD3
SCHEMBL4050835 0.82 DRD2 (0.39) CYP51A1DRD2PYGLSTAT6TAS1R3
SCHEMBL4052196 0.82 DRD4 (0.38) CYP51A1DRD2PYGLSTAT6DRD3
SCHEMBL7997110 0.82 DRD2 (0.38) CYP51A1DRD2PYGLSTAT6DRD3
SCHEMBL19856857 0.81 DRD2 (0.39) CYP51A1DRD2PYGLSTAT6DRD3
SCHEMBL19856858 0.81 DRD2 (0.39) CYP51A1DRD2PYGLSTAT6DRD3
SCHEMBL4056098 0.81 DRD2 (0.35) CYP51A1DRD2PYGLSTAT6

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2009111680-A1 TRPV4 ANTAGONISTS SMITHLINE BEECHAM CORPORATION (US) 2009-09-11 WO disclosed