SCHEMBL7998218

SCHEMBL7998218

Cc1c(Cn2ccnc2[N+](=O)[O-])cccc1NC(=O)OC(C)(C)C

nearest known ligand 0.46

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
SLC29A1 Q99808 1/20 0.46
CYP3A4 P08684 1/20 0.40
CYP2D6 P10635 1/20 0.40
OPRK1 P41145 1/20 0.40
P2RX7 Q99572 1/20 0.40
CA12 O43570 4/20 0.39
CA1 P00915 4/20 0.39
CA2 P00918 4/20 0.39
CA9 Q16790 4/20 0.39
LMNA P02545 1/20 0.38
THRB P10828 1/20 0.38
CYP2C19 P33261 1/20 0.38
SMN1; SMN2 Q16637 2/20 0.38
TYMP P19971 3/20 0.36
METAP1 P53582 1/20 0.36
BRD4 O60885 2/20 0.36
GPR139 Q6DWJ6 1/20 0.35
KMT2A Q03164 1/20 0.35
BRD9 Q9H8M2 1/20 0.35
NPC1 O15118 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7983853 0.93 SLC29A1 (0.41) SLC29A1CYP3A4CYP2D6OPRK1P2RX7
SCHEMBL7983855 0.85 SLC29A1 (0.36) SLC29A1CYP3A4CYP2D6OPRK1P2RX7
SCHEMBL7983856 0.82 P2RX7 (0.39) SLC29A1CYP3A4CYP2D6OPRK1P2RX7
SCHEMBL7983691 0.77 LMNA (0.38) SLC29A1CYP3A4CYP2D6OPRK1CA12
SCHEMBL7996398 0.77 CYP3A4 (0.40) CYP3A4CYP2D6OPRK1CA12CA1
SCHEMBL7998436 0.76 CYP3A4 (0.42) CYP3A4CYP2D6OPRK1CA12CA1
SCHEMBL7998028 0.75 TBXAS1 (0.48) P2RX7BRD4BRD9
SCHEMBL7984571 0.74 CYP3A4 (0.43) CYP3A4CYP2D6OPRK1CA12CA1
SCHEMBL8001778 0.73 F2 (0.33) CYP3A4CYP2D6OPRK1CA12CA1
SCHEMBL8001605 0.73 LMNA (0.42) CYP3A4CYP2D6OPRK1CA12CA1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2001034578-A1 COMPOUNDS WITH ANTI-HELICOBACTER PYLORI ACTIVITY ASTRAZENECA AB (SE) 2001-05-17 WO disclosed