SCHEMBL8002260

SCHEMBL8002260

Cn1c(C(F)(F)F)cc(=O)n(-c2ccc(C#N)c(S(=O)(=O)Cl)c2)c1=O

nearest known ligand 0.38

Predicted protein targets (top 6)

geneUniProtsupporting neighboursconfidence
AR P10275 14/20 0.38
TRPV4 Q9HBA0 1/20 0.36
BCAT2 O15382 1/20 0.36
BCAT1 P54687 1/20 0.36
NR1H2 P55055 2/20 0.34
NR1H3 Q13133 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3555928 0.84 TSHR (0.34) AR
SCHEMBL1574267 0.81 AR (0.38) ARBCAT2BCAT1
SCHEMBL8465633 0.81 AR (0.37) ARBCAT2BCAT1
SCHEMBL8190792 0.79 AR (0.39) ARBCAT2BCAT1
SCHEMBL8464476 0.78 AR (0.39) ARBCAT2BCAT1
SCHEMBL6920290 0.78 VCAM1 (0.41) ARBCAT2BCAT1
SCHEMBL9469308 0.76 POLB (0.41) ARBCAT2BCAT1
SCHEMBL3545755 0.76 MMP2 (0.36)
SCHEMBL8936370 0.74 MEN1 (0.39)
SCHEMBL8936415 0.74 GSTO1 (0.41)

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6107252-A 1-((3-AMINOSULFONYL,4-CYANO,6-SUBSTITUTED PHENYL)-),3,4,5-SUBSTITUTED-1,2,3,6-TETRAHYDROPYRIMIDIN-2,6-DIONE COMPOUNDS; HERBICIDAL ACTIVITY AND AT THE SAME TIME COMPATIBILITY WITH CROP PLANTS BAYER AKTIENGESELLSCHAFT (DE) 2000-08-22 US disclosed